Membrane transporter-Others

Cat.No.	Product Name	Information	Area
T4595	YHO-13177	YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of...	Cancer
T4610	BMS-927711	BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor a...	Migraine
T4590	L-KAWAIN	Kawain is one of the six major kavalactones found in the Piper methysticum (kava) pla...
T2S2335	Dehydroevodiamine	Dehydroevodiamine, a constituent of Evodia rutaecarpa, has various biological effects...
T1125	(+)-Shikonin	Shikonin is an TMEM16A chloride channel inhibitor (IC50: 6.5 μM). Shikonin is also a ...
T4363	CGP 52432	CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
T4190	Ticlopidine	Ticlopidine is an antiplatelet drug in the thienopyridine family which is an adenosin...	Ischaemia; Thromboembolism
T4054	Dantrolene sodium hemiheptahydrate	Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to...	Immunology
T4030	ML213	ML213 is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhance...	Others
T3994	Verinurad	Verinurad (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for t...	Metabolism
T3528	Senicapoc	Senicapoc is a potent inhibitor of the Gardos channel and ameliorates RBC dehydration...	Others
T3959	ICA069673	ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).	Others
T3534	TETRABENAZINE	Tetrabenazine (Racemate) is a selective and reversible inhibitor of vesicular monoami...	Nervous system
T3581	KS176	KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BC...	Others
T3690	A 740003	A 740003 is an effective and specific P2X7?receptor antagonist (IC50: 18/40 nM, for r...	Immunology
T3639	A-804598	A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9...	Others
T3093	Spermine?Tetrahydrochloride	Spermine is a polyamine involved in cellular metabolism found in all eukaryotic cells...	Other
T3210	AZD-3965	AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1).	Cancer
T2657	Elacridar	Elacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.	Other
T2486	IOWH-032	IOWH032, a synthetic CFTR inhibitor, has been investigated for the treatment of chol...	Cancer
T2257	AdipoRon	AdipoRon is an orally bioavailable adiponectin receptor agonist. It can combine with ...	Other
T2196	Fipronil	Fipronil is a broad-use insecticide that belongs to the phenylpyrazole chemical famil...	Immunology
T1768	7ACC2	7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for [14C]-lactate influx; new ...	Other
T1672	Dimesna	Dimesna is a synthetic derivative of dithio-ethane sulfonate with uroprotective prope...	Immunology
T1479	Isosorbide dinitrate	Isosorbide dinitrate is a vasodilator used in the treatment of angina pectoris.	Cardiovascular System
T1410	Torasemide	Torsemide is an anilinopyridine sulfonylurea belonging to the class of loop diuretics...	Cardiovascular System
T0837	Furosemide	Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chron...	Cardiovascular System
T0715	Chlormezanone	Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It h...	Nervous system
T0490	Chlorpropamide	Chlorpropamide is a sulfonylurea hypoglycemic agent used in the treatment of non-insu...	Metabolism system
T0295	Digitoxin	Digitoxin is an effective Na+/K+-ATPase inhibitor (EC50 value: 0.78 μM).	Cardiovascular System

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