Cat.No. |
Product Name |
Information |
Area |
T4595 |
YHO-13177 |
YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of... |
Cancer |
T4610 |
BMS-927711 |
BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor a... |
Migraine |
T4590 |
L-KAWAIN |
Kawain is one of the six major kavalactones found in the Piper methysticum (kava) pla... |
|
T2S2335 |
Dehydroevodiamine |
Dehydroevodiamine, a constituent of Evodia rutaecarpa, has various biological effects... |
|
T1125 |
(+)-Shikonin |
Shikonin is an TMEM16A chloride channel inhibitor (IC50: 6.5 μM). Shikonin is also a ... |
|
T4363 |
CGP 52432 |
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM). |
|
T4190 |
Ticlopidine |
Ticlopidine is an antiplatelet drug in the thienopyridine family which is an adenosin... |
Ischaemia; Thromboembolism |
T4054 |
Dantrolene sodium hemiheptahydrate |
Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to... |
Immunology |
T4030 |
ML213 |
ML213 is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhance... |
Others |
T3994 |
Verinurad |
Verinurad (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for t... |
Metabolism |
T3528 |
Senicapoc |
Senicapoc is a potent inhibitor of the Gardos channel and ameliorates RBC dehydration... |
Others |
T3959 |
ICA069673 |
ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM). |
Others |
T3534 |
TETRABENAZINE |
Tetrabenazine (Racemate) is a selective and reversible inhibitor of vesicular monoami... |
Nervous system |
T3581 |
KS176 |
KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BC... |
Others |
T3690 |
A 740003 |
A 740003 is an effective and specific P2X7?receptor antagonist (IC50: 18/40 nM, for r... |
Immunology |
T3639 |
A-804598 |
A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9... |
Others |
T3093 |
Spermine?Tetrahydrochloride |
Spermine is a polyamine involved in cellular metabolism found in all eukaryotic cells... |
Other |
T3210 |
AZD-3965 |
AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1). |
Cancer |
T2657 |
Elacridar |
Elacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor. |
Other |
T2486 |
IOWH-032 |
IOWH032, a synthetic CFTR inhibitor, has been investigated for the treatment of chol... |
Cancer |
T2257 |
AdipoRon |
AdipoRon is an orally bioavailable adiponectin receptor agonist. It can combine with ... |
Other |
T2196 |
Fipronil |
Fipronil is a broad-use insecticide that belongs to the phenylpyrazole chemical famil... |
Immunology |
T1768 |
7ACC2 |
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for [14C]-lactate influx; new ... |
Other |
T1672 |
Dimesna |
Dimesna is a synthetic derivative of dithio-ethane sulfonate with uroprotective prope... |
Immunology |
T1479 |
Isosorbide dinitrate |
Isosorbide dinitrate is a vasodilator used in the treatment of angina pectoris. |
Cardiovascular System |
T1410 |
Torasemide |
Torsemide is an anilinopyridine sulfonylurea belonging to the class of loop diuretics... |
Cardiovascular System |
T0837 |
Furosemide |
Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chron... |
Cardiovascular System |
T0715 |
Chlormezanone |
Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It h... |
Nervous system |
T0490 |
Chlorpropamide |
Chlorpropamide is a sulfonylurea hypoglycemic agent used in the treatment of non-insu... |
Metabolism system |
T0295 |
Digitoxin |
Digitoxin is an effective Na+/K+-ATPase inhibitor (EC50 value: 0.78 μM). |
Cardiovascular System |