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Membrane transporter-Others
Cat.No. Product Name Information Area
T5102 TGN020 TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water ... Others
T4595 YHO-13177 YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of... Cancer
T4610 BMS-927711 BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor a... Migraine
T4590 L-KAWAIN Kawain is one of the six major kavalactones found in the Piper methysticum (kava) pla...
T2S2335 Dehydroevodiamine Dehydroevodiamine, a constituent of Evodia rutaecarpa, has various biological effects...
T1125 (+)-Shikonin Shikonin is an TMEM16A chloride channel inhibitor (IC50: 6.5 μM). Shikonin is also a ...
T4363 CGP 52432 CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
T4190 Ticlopidine Ticlopidine is an antiplatelet drug in the thienopyridine family which is an adenosin... Ischaemia; Thromboembolism
T4054 Dantrolene sodium hemiheptahydrate Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to... Immunology
T4030 ML213 ML213 is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhance... Others
T3994 Verinurad Verinurad (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for t... Metabolism
T3528 Senicapoc Senicapoc is a potent inhibitor of the Gardos channel and ameliorates RBC dehydration... Others
T3959 ICA069673 ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM). Others
T3534 TETRABENAZINE Tetrabenazine (Racemate) is a selective and reversible inhibitor of vesicular monoami... Nervous system
T3581 KS176 KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BC... Others
T3690 A 740003 A 740003 is an effective and specific P2X7?receptor antagonist (IC50: 18/40 nM, for r... Immunology
T3639 A-804598 A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9... Others
T3093 Spermine?Tetrahydrochloride Spermine is a polyamine involved in cellular metabolism found in all eukaryotic cells... Other
T3210 AZD-3965 AZD3965 is a selective inhibitor of monocarboxylate transporter 1 (MCT1). Cancer
T2657 Elacridar Elacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor. Other
T2486 IOWH-032 IOWH032, a synthetic CFTR inhibitor, has been investigated for the treatment of chol... Cancer
T2257 AdipoRon AdipoRon is an orally bioavailable adiponectin receptor agonist. It can combine with ... Other
T2196 Fipronil Fipronil is a broad-use insecticide that belongs to the phenylpyrazole chemical famil... Immunology
T1768 7ACC2 7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for [14C]-lactate influx; new ... Other
T1672 Dimesna Dimesna is a synthetic derivative of dithio-ethane sulfonate with uroprotective prope... Immunology
T1479 Isosorbide dinitrate Isosorbide dinitrate is a vasodilator used in the treatment of angina pectoris. Cardiovascular System
T1410 Torasemide Torsemide is an anilinopyridine sulfonylurea belonging to the class of loop diuretics... Cardiovascular System
T0837 Furosemide Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chron... Cardiovascular System
T0715 Chlormezanone Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It h... Nervous system
T0490 Chlorpropamide Chlorpropamide is a sulfonylurea hypoglycemic agent used in the treatment of non-insu... Metabolism system