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Results for "

thz-1

" in TargetMol Product Catalog

Inhibitors & Agonists
6

THZ1

THZ1 2HCl, CDK7 inhibitor

T36641604810-83-4

THZ1 (CDK7 inhibitor) is a selective covalent inhibitor of CDK7, exhibiting binding affinity to the cysteine residue located at the outer end of the classical kinase domain, thus conferring high selectivity for CDK7, with an IC50 of 3.2 nM.

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THZ2

CDK7-IN-1

T72961604810-84-5

THZ2 (CDK7-IN-1), an analog of THZ1, is a potent and selective CDK7 inhibitor(IC50:13.9 nM),with the potential to treat Triple-negative breast cancer (TNBC).

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bio-THZ1

T105461604811-14-4

bio-THZ1 is a biotinylated version of THZ1, a selective and irreversibly covalent CDK7 inhibitor (IC50: 3.2 nM).

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THZ1-R

T131531621523-07-6

THZ1-R displays diminished activity for CDK7 inhibition(Kd:142 nM).

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6-8 weeks

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(E/Z)-THZ1 2HCl

(E Z)-THZ1 2HCl, (E Z)-THZ1 Dihydrochloride

T353322095433-94-4

THZ1 2HCl (THZ1 Dihydrochloride) is a selective, covalent, and allosteric inhibitor of CDK7 with an IC50 of 3.2 nM. THZ1 2HCl has antiproliferative effects on a variety of cancer cell lines.

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THZ-P1-2

T394592058075-45-7

THZ-P1-2 is a selective and potent PI5P4K inhibitor with anti-leukemic activity that acts by disrupting mitochondrial homeostasis and autophagy.THZ-P1-2 induces cell death and mitochondrial damage, and can be used in the study of leukemias.

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7-10 days

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