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ibet-bd1

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
GSK778
T97032451862-42-1
GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1 (IC50s = 75 nM), BRD3 BD1 (IC50s = 41 nM), BRD4 BD1 (IC50s = 41 nM), and BRDT BD1 (IC50s = 143 nM). GSK778 inhibits proliferation, induces a cell cycle arrest and apoptosis.
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7-10 days
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