Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
Applied FilterClear all
TargetMol | Tags By Target
  • CDK
    (1)
  • Calcium Channel
    (1)
  • GPCR19
    (1)
  • TRP/TRPV Channel
    (1)
Filter
Search Result
Results for "

ca2+ channel agonist 1

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    4
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    1
    TargetMol | Peptide_Products
Ca2+ channel agonist 1
T106591402821-24-2
Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for motor nerve terminal dysfunction.
  • Inquiry Price
Size
QTY
TargetMol | Inhibitor Sale
TRPV4 agonist-1
T132142314467-60-0
TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).
  • Inquiry Price
1-2 weeks
Size
QTY
TGR5 Receptor Agonist
T18241197300-24-5
TGR5 is a potent TGR5(GPCR19) agonist.
  • Inquiry Price
Size
QTY
TargetMol | Inhibitor Sale
CALP1 TFA
T75791
CALP1 TFA, a calmodulin (CaM) agonist with a dissociation constant (Kd) of 88 µM, selectively binds to the CaM EF-hand Ca2+-binding site, inhibiting calcium channel opening. This action blocks calcium influx and apoptosis with an IC50 of 44.78 µM, modulates glutamate receptor channel activity, and impedes a store-operated nonselective cation channel. Additionally, CALP1 TFA enhances CaM-dependent phosphodiesterase activity, denoting its multifaceted role in modulating cellular calcium dynamics [1] [2] [3] [4].
  • Inquiry Price
Size
QTY