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T4610

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  • Inhibitors & Agonists
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Rimegepant
BMS-927711, BMS927711, BMS 927711, BHV-3000
T46101289023-67-1
Rimegepant (BMS 927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
  • $46
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Rimegepant sulfate hydrate
T708371374024-48-2
Rimegepant, also known as BMS-927711 and BHV-3000, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist in clinical trials for treating migraines. Rimegepant has shown in vivo efficacy without vasoconstriction effect. BMS-927711 is superior to placebo at several different doses (75 mg, 150 mg, and 300 mg) and has an excellent tolerability profile.
  • $2,870
10-14 weeks
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Rimegepant hemisulfate
BMS-927711 hemisulfate, BHV-3000 hemisulfate
T2143451642783-82-1
Rimegepant (BMS-927711) hemisulfate is a potent, orally active selective competitive antagonist of the calcitonin gene-related peptide (CGRP) receptor, with a Ki of 0.027 nM and an IC50 of 0.14 nM for the hCGRP receptor. Rimegepant hemisulfate is utilized in migraine research.
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