T1051

Retinoic acid (Tretinoin), a metabolite of vitamin A, is a natural agonist of the retinoic acid receptor RAR and inhibits RARα/β/γ (IC50=14 nM). Retinoic acid induces cellular differentiation, reduces cellular proliferation, and inhibits tumorigenesis.

Prenyl-IN-1 is a potent and selective prenylation inhibitor of geranylgeranyltransferase or farnesyltransferase.Prenyl-IN-1 shows anti-oxidative stress effects in a Parkinson's model. Prenyl-IN-1 showed anti-oxidative stress in a Parkinson's model.

CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, and gastrointestinal disorders, psychosis, and cardiovascular.

Anti-hypertensive sulfonanilide 1 is an antihypertensive compound.

Benzothiohydrazide is an analog of isoniazid with anti-tuberculosis activity and can be used to isolate fungi and bacteria.

FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).

Anti-Heart Failure Agent 1 is an orally available compound suitable for treating heart failure without causing vomiting, nausea, or restlessness.

Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).

The S-enantiomer of BET-BAY 002, referred to as BET-BAY 002 S enantiomer, is a potent inhibitor of BET (Bromodomain and Extra-Terminal motif proteins).

BET-BAY 002 is an effective BET bromodomain inhibitor demonstrating efficacy in vivo and in vitro against multiple myeloma and leukaemia models.

Retinoic acid-D5 is the deuterium-labeled form of Retinoic acid. Retinoic acid (T1051) is a natural RAR receptor agonist with an IC50 of 14 nM for RARα/β/γ and a Kd of 17 nM for PPARβ/δ. Retinoic acid, a metabolite of vitamin A, plays an important role in cell growth, differentiation and organ development. Retinoic acid (T1051) acts by activating retinoic acid receptor alpha as an inhibitor of the transcription factor Nrf2.

Retinoic acid-D6 is the deuterated form of Retinoic acid. Retinoic acid, a metabolite of vitamin A, plays a crucial role in cell growth, differentiation, and organ development. It is a natural agonist of the RAR nuclear receptor, with an IC50 of 14 nM for RARα/β/γ, and has a Kd value of 17 nM when binding to PPARβ/δ. Additionally, Retinoic acid (T1051) can inhibit the transcription factor Nrf2 by activating retinoic acid receptors.