arm1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T21859	ARM1		Aminopeptidase , Epoxide Hydrolase
	ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.		Aminopeptidase , Epoxide Hydrolase
T10682L	CARM1-IN-1	CARM1-IN-7G	Histone Methyltransferase
	CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM.		Histone Methyltransferase
T60908	SARM1-IN-2		Others
	SARM1-IN-2 is a potent SARM1 inhibitor for the study of metabolic and neurological related diseases.		Others
T63180	CARM1-IN-3 dihydrochloride
	CARM1-IN-3 dihydrochloride (compound 17b) CARM1-IN-3 dihydrochloride (compound 17b) is a potent, selective coactivator-associated arginine methyltransferase (CARM1) inhibitor that acts on CARM1 (IC50: 0.07 μM) and CARM3 ...
T64186	CARM1-IN-1 hydrochloride
	CARM1-IN-1 hydrochloride is a potent and selective inhibitor of CARM1 (IC50: 8.6 μM) with low inhibition of PRMT1 and SET7.
T79007	CARM1-IN-3		Histone Methyltransferase
	CARM1-IN-3 (compound 17b) is a potent, selective inhibitor of co-activator associated arginine methyltransferase (CARM1), exhibiting IC50 values of 0.07 µM for CARM1 and greater than 25 µM for CARM3 [1].		Histone Methyltransferase
T79742	CARM1 degrader-2		Histone Methyltransferase
	PROTAC CARM1 degrader-2 (compound 3e), with a DC50 value of 8.8 nM, is a VHL- and proteasome-dependent degrader of co-activator associated argininemethyltransferase (CARM1). It not only promotes the degradation of CARM1 ...		Histone Methyltransferase
T79741	CARM1 degrader-1		Histone Methyltransferase
	PROTAC CARM1 degrader-1 (compound 3b) serves as a highly potent degrader (DC50=8.1 nM) of the co-activator associated arginine methyltransferase (CARM1). This compound facilitates the degradation of CARM1 via the VHL-pro...		Histone Methyltransferase

Compounds

ARM1

T21859

Synonym:

Target: Aminopeptidase, Epoxide Hydrolase

CARM1-IN-1

T10682L

Synonym: CARM1-IN-7G

Target: Histone Methyltransferase

CARM1-IN-3 dihydrochloride

T63180

Synonym:

Target:

CARM1-IN-1 hydrochloride

Target: Histone Methyltransferase

CARM1 degrader-2

T79742

Synonym:

Target: Histone Methyltransferase

CARM1 degrader-1

T79741

Synonym:

Target: Histone Methyltransferase

Recombinant Proteins

Species：

Expression System：

Tag：

Cat No.	Product Name	Species	Expression System
TMPY-01900	Kallikrein 4/KLK4 Protein, Human, Recombinant (His)	Human	HEK293
	Kallikrein-4, also known as Enamel matrix serine proteinase 1, Kallikrein-like protein 1, KLK-L1, Serine protease 17, KLK4, PRSS17, and EMSP1, is a secreted protein that belongs to the peptidase S1 family and Kallikrein ...
TMPH-01740	SARM1 Protein, Human, Recombinant (His & Myc)	Human	Baculovirus
	NAD(+) hydrolase, which plays a key role in axonal degeneration following injury by regulating NAD(+) metabolism. Acts as a negative regulator of MYD88- and TRIF-dependent toll-like receptor signaling pathway by promotin...
TMPH-01741	SARM1 Protein, Human, Recombinant (His & KSI)	Human	E. coli
	NAD(+) hydrolase, which plays a key role in axonal degeneration following injury by regulating NAD(+) metabolism. Acts as a negative regulator of MYD88- and TRIF-dependent toll-like receptor signaling pathway by promotin...