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(1)
By Target- CDK
- ERK(1)
- ROCK(1)
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By Target By ResearchField- Cancer(1)
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Results for "
pt-262
" in TargetMol Product Catalog- Inhibitors & Agonists1
PT-262
PT262, PT 262
T2846986811-36-1
PT-262 is a potent Rho-associated protein kinase (ROCK) inhibitor with an IC50 value of approximately 5 μM, and it induces mitochondrial membrane potential loss, enhances caspase-3 activation, and promotes apoptosis, while concurrently inhibiting ERK and CDC2 phosphorylation through a p53-independent signaling pathway, disrupting cytoskeletal organization and cell migration, and collectively exerting broad anticancer activity that makes PT-262 a valuable tool for mechanistic cancer biology and signal transduction research.
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