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Results for "

cbp brd

" in TargetMol Product Catalog

Inhibitors & Agonists
6

Pocenbrodib

P-300, FT-7051

T696912304372-79-8In house

Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP p300 family with potential antitumour activity and is palatable for cancer research.

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10-14 weeks

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SGC-CBP30

T66681613695-14-9

SGC-CBP30 is an effective CREBBP EP300 inhibitor (IC50: 21 38 nM).

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Cited

l-moses dihydrochloride

T62424

L-Moses (L-45) dihydrochloride is the first potent and selective inhibitor of the p300 CBP-associated factor (PCAF) bromodomain (Brd) with a dissociation constant (Kd) of 126 nM.

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10-14 weeks

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L-Moses

L-45

T11796L2079885-05-3

L-45 is the first potent and cell-active bromodomain (Brd) inhibitor of p300 CBP-associated factor (PCAF) (Kd: 126±15 nM).

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8-10 weeks

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EP300/CBP-IN-1

T863772638507-71-6

EP300 CBP-IN-1 (compound 172), a potent inhibitor of EP300 CBP, exhibits IC 50 values of 2.1 nM for EP300 BRD and 2.3 nM for CBP BRD. It effectively inhibits the proliferation of prostate cancer CWR22RV1 cells [1].

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10-14 weeks

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MS417

GTPL7512

T16154916489-36-6

MS417 (GTPL7512) is an inhibitor of BET-specific BRD4(BRD4-BD1 and BRD4-BD2 with IC50s of 30, 46 nM and Kds of 36.1, 25.4 nM, respectively), with weak selectivity at CBP BRD with IC50 of 32.7 μM.

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