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Search Result

Search Results for " p-450 "

Targets

Aromatase

26

Compounds

3

Natural Products

Cat No. Product Name Synonyms Targets
T7556 Fadrozole hydrochloride CGS 16949A Aromatase
Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that has been shown to suppress estrogen production in the ovaries of fish.
T25283 Cytochrome P450 2C9 Cyp2C9,Human cytochrome P450 2C9,Cytochrome P 450 2C9,S-Mephenytoin 4-hydroxylase
Cytochrome P450 2C9 is a cytochrome P-450 subtype that possesses specificity for acidic xenobiotics. It oxidizes a wide range of important clinical drugs under the categories of nonsteroidal anti-inflammatory agents, ant...
TP2238 Cytochrome P450 CYP1B1 (190-198) [Homo sapiens] Others
Cytochrome P450 CYP1B1 (190-198) [Homo sapiens] is a small heme protein found loosely associated with the inner membrane of the mitochondrion.
T117521 7-BFC 7-Benzyloxy-4-(trifluoromethyl)coumarin,Y040-0031 P450
7-BFC (7-Benzyloxy-4-(trifluoromethyl)coumarin) is a coumarin-like fluorescent substrate that serves as a biomarker for cytochrome P 450 and can be used to study CYP isoforms and cytochrome P 450 metabolism.
T1597 Proadifen hydrochloride U-5446,RP-5171,SKF-525A P450
Proadifen hydrochloride (RP-5171) is an inhibitor of drug metabolism and cytochrome P-450 enzyme system activity.
T1378 Tegafur Fluorafur,FT-207,NSC 148958,FT 207 Nucleoside Antimetabolite/Analog , DNA/RNA Synthesis
Tegafur (FT 207) is a congener of the antimetabolite fluorouracil with antineoplastic activity. Tegafur is a prodrug that is gradually converted to fluorouracil in the liver by the cytochrome P-450 enzyme.
T27918 LY 43578 LY-43578,LY43578 P450 , Aromatase
LY 43578 is an orally active aromatase inhibitor. LY43578 could inhibit O-demethylation of P-450-dependent p-nitroanisole and N-demethylation of ethylmorphine (IC50 of 0.3 and 5 μm, respectively) in rat liver microsomes....
T0120 Voriconazole UK-109496 Antifection , Antifungal
Voriconazole (UK-109496) is a triazole antifungal agent that specifically inhibits STEROL 14-ALPHA-DEMETHYLASE and CYTOCHROME P-450 CYP3A.
T7696 3-Cyano-7-ethoxycoumarin Others
3-Cyano-7-ethoxycoumarin is cytochrome P450 (CYP) isoforms CYP1A1 and CYP1A2 .
T6686 Sulconazole mononitrate Exelderm,Sulconazole Nitrate,RS 44872 Antibacterial , Antibiotic , Antifungal
Sulconazole mononitrate (Exelderm) is the nitrate salt form of sulconazole, a synthetic imidazole derivative with the antifungal property. Sulconazole mononitrate inhibits fungal cytochrome P-450 sterol C-14 alpha-demeth...
T5952 Diniconazole Rac-diniconazole Antibacterial
Diniconazole (Rac-diniconazole) is a fungicide. It is known as a plant hormone abscisic acid (ABA) catabolic inhibitor, and acts as a potent competitive inhibitor of recombinant Arabidopsis ABA 8'-hydroxylase, CYP707A3.
T0922 Zoxazolamine NSC 24995,Contrazole Others
Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant. Zoxazolamine acts centrally as a muscle relaxant, but the mechanism of its action is not understood.
T22229 Acid Yellow 36 Metanil Yellow Others
Acid Yellow 36 (Metanil Yellow) is an azo dye and a pH indicator. Acid Yellow 36 changes its color from red at pH 1.2 to yellow at pH 2.3.
T33110 M 79193 M79193,M-79193
M 79193 induces total hepatic microsomal cytochrome P-450.
T34990 UK 39671
UK 39671 is an inhibitor of cytochrome P-450(CAM) inhibitor.
T25591 Lab 170250F Lab-170250F,Lab170250F
Lab 170250F is a potent cytochrome P-450-obtusifoliol-14-demethylase inhibitor.
T69553 p,p'-DDMS
p,p'-DDMS is a water soluble and highly specific inhibitor of cytochrome P-450 omega-hydroxylase.
T31815 Flumecinol Zyxorin
Flumecinol is a hepatic enzyme (cytochrome P-450 monooxygenases) inducer.
T69167 Buthiobate
Buthiobate is a fungicide which inhibits lanosterol 14 alpha-demethylation catalyzed by a cytochrome P-450.
T19553 RPR132595A NPC Others
RPR132595A is an active CPT-11 metabolite, it is generated by cytochrome P-450 3A4 (CYP3A4).
T78069 RPR132595A hydrochloride NPC hydrochloride Drug Metabolite
RPR132595A (NPC) hydrochloride, an active metabolite of CPT-11, is produced via cytochrome P-450 3A4 (CYP3A4) metabolism and is ultimately eliminated via urinary excretion [1].
T78135 Nicotelline Nicotellin
Nicotelline, also known as Nicotellin, is an alkaloid associated with nicotine and acts as a modest inhibitor of the enzyme human cDNA-expressed cytochrome P-450 2A6 (CYP2A6), which is responsible for coumarin 7-hydroxyl...
T36666 Dehydro Warfarin
Dehydro warfarin is a metabolite of (±)-warfarin .1It is formed from (±)-warfarin by rat liver microsomes. 1.Kaminsky, L.S., Fasco, M.J., and Guengerich, F.P.Comparison of different forms of liver, kidney, and lung micro...
T61259 Valganciclovir
Valganciclovir, the L-valyl ester of ganciclovir, is a prodrug effectively converted to ganciclovir in the body, serving as an antiviral medication for cytomegalovirus (CMV) infections. In vitro studies demonstrate that ...
T38269 Purfalcamine
Purfalcamine is an orally active, selective Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1) inhibitor with an IC50 of 17 nM and an EC50 of 230 nM. Purfalcamine has antimalarial activity and causes mala...
T35463 (±)14(15)-EET (±)14,15-EET,(±)14,15-EpETrE,(±)14(15)-EET
(±)14(15)-EET is a metabolite of arachidonic acid that is formed via epoxidation of arachidonic acid by cytochrome P450.[1],[2] It prevents increases in leukotriene B4, ICAM-1, and chemokine (C-C motif) ligand 1 (CCL2) i...

Compounds

Fadrozole hydrochloride
T7556
Synonym: CGS 16949A
Target: Aromatase
Cytochrome P450 2C9
T25283
Synonym: Cyp2C9,Human cytochrome P450 2C9,Cytochrome P 450 2C9,S-Mephenytoin 4-hydroxylase
Target:
Cytochrome P450 CYP1B1 (190-198) [Homo sapiens]
TP2238
Synonym:
Target: Others
7-BFC
T117521
Synonym: 7-Benzyloxy-4-(trifluoromethyl)coumarin,Y040-0031
Target: P450
Proadifen hydrochloride
T1597
Synonym: U-5446,RP-5171,SKF-525A
Target: P450
Tegafur
T1378
Synonym: Fluorafur,FT-207,NSC 148958,FT 207
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
LY 43578
T27918
Synonym: LY-43578,LY43578
Target: P450, Aromatase
Voriconazole
T0120
Synonym: UK-109496
Target: Antifection, Antifungal
3-Cyano-7-ethoxycoumarin
T7696
Synonym:
Target: Others
Sulconazole mononitrate
T6686
Synonym: Exelderm,Sulconazole Nitrate,RS 44872
Target: Antibacterial, Antibiotic, Antifungal
Diniconazole
T5952
Synonym: Rac-diniconazole
Target: Antibacterial
Zoxazolamine
T0922
Synonym: NSC 24995,Contrazole
Target: Others
Acid Yellow 36
T22229
Synonym: Metanil Yellow
Target: Others
M 79193
T33110
Synonym: M79193,M-79193
Target:
UK 39671
T34990
Synonym:
Target:
Lab 170250F
T25591
Synonym: Lab-170250F,Lab170250F
Target:
p,p'-DDMS
T69553
Synonym:
Target:
Flumecinol
T31815
Synonym: Zyxorin
Target:
Buthiobate
T69167
Synonym:
Target:
RPR132595A
T19553
Synonym: NPC
Target: Others
RPR132595A hydrochloride
T78069
Synonym: NPC hydrochloride
Target: Drug Metabolite
Nicotelline
T78135
Synonym: Nicotellin
Target:
Dehydro Warfarin
T36666
Synonym:
Target:
Valganciclovir
T61259
Synonym:
Target:
Purfalcamine
T38269
Synonym:
Target:
(±)14(15)-EET
T35463
Synonym: (±)14,15-EET,(±)14,15-EpETrE,(±)14(15)-EET
Target:
Cat No. Product Name Synonyms Targets
TN1078 Seneciphylline P450 , GST
Seneciphylline, one of the hepatotoxic pyrolizidine alkaloids, has mutagenic activity in Drosophila and their transfer into rat milk.Seneciphylline can significantly increased the activities of epoxide hydrase and glutat...
T1011 Itraconazole R51211 P450 , Hedgehog/Smoothened , Antibiotic , Autophagy , Antifungal
Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis.
T40859 5-Hydroxy-8-methoxypsoralen 5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen
5-Hydroxy-8-methoxypsoralen (5-Hydroxyxanthotoxin) is a metabolite derived from Xanthotoxin, which acts as a potent tricyclic furocoumarin suicide inhibitor of CYP (cytochrome P-450). It is employed as an agent for the t...

Natural Products

Seneciphylline
TN1078
Synonym:
Target: P450, GST
Itraconazole
T1011
Synonym: R51211
Target: P450, Hedgehog/Smoothened, Antibiotic, Autophagy, Antifungal
5-Hydroxy-8-methoxypsoralen
T40859
Synonym: 5-Hydroxyxanthotoxin,5-Hydroxy-8-methoxypsoralen
Target:
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