Home Tools
Log in
Cart

Search Result

Search Results for " eris "

Targets

38

Compounds

11

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T13015 STING agonist-4 STING
STING agonist-4 is an agonist of stimulator of Interferon Genes (STING) receptor(IC50 of 20 nM).
T13613 ChX710 STING
ChX710 activates the type I interferon response to cytosolic DNA by priming specific Interferon-Stimulated Genes (ISGs), inducing the ISRE promoter sequence, and facilitating the phosphorylation of Interferon Regulatory ...
T7329 C-178 STING
C-178 is a covalent inhibitor of STING, binds to Cys91 on STING to block its palmitoylation and prevents recruitment and phosphorylation of TBK1 in HEK293T cells.
T9853 STING activator Compound 53 STING
STING activator Compound 53 based on an oxindole core structure demonstrated robust on-target functional activation of STING (human EC50 185 nM) in immortalised and primary cells and a cytokine induction fingerprint cons...
T6919 Omaveloxolone RTA-408 Apoptosis , Others , Nrf2 , STING
Omaveloxolone (RTA-408) (RTA-408) is a synthetic triterpenoid that activates the cytoprotective transcription factor Nrf2 and inhibits NF-κB signaling. Phase 2.
T9554 SN-008 STING
SN-008 is a less active analog SN-011 which is a STING antagonist. SN-008 can be used as a negative control.
T5674 H-151 STING
H-151 is a highly potent and selective STING antagonist. H-151 covalently binds to Cys91 of STING and inhibits palmitoylation of Cys91, thereby inhibiting STING activity. H-151 can be used in the study of autoinflammator...
T8655 SR-717 STING
SR-717 is a cGAMP analog, a non-nucleoside STING agonist that induces a "closed" activation conformation of STING. SR-717 has antitumor activity and promotes activation of immune cells and cross-presentation of antigens.
T8798 MSA-2 STING
MSA-2 is a potent and orally available non-nucleotide STING agonist.
T9029 STING-IN-3 C-171 STING
STING-IN-3 (C-171) is an inhibitor of stimulator of interferon genes (STING). It binds to STING, inhibits its palmitoylation, and prevents the recruitment and phosphorylation of TBK1.
T5154 C-176 C176,STING inhibitor 1 STING
C-176 (STING inhibitor 1) is a strong, covalent mouse STING inhibitor
T5516 DiABZI STING agonist-1 trihydrochloride STING
diABZI STING agonist-1 (trihydrochloride) is stimulator of interferon genes (STING) receptor agonist.
T8328 STING agonist-1 G10 Virus Protease , STING
STING agonist-1 (G10) is a human-specific STING agonist,elicits antiviral activity against emerging Alphaviruses.
T9028 STING-IN-2 C-170 STING
STING-IN-2 (C-170) is a potent and covalent inhibitor of STING. C-170 efficiently inhibits both mouse STING (mmSTING) and human STING (hsSTING). It can be used for autoinflammatory disease research.
T7081 CCCP Carbonyl Cyanide m-Chlorophenylhydrazone,Carbonyl cyanide 3-chlorophenylhydrazone Apoptosis , IκB/IKK , COX , Mitochondrial Metabolism , STING , IFNAR , Antibacterial
CCCP (Carbonyl Cyanide m-Chlorophenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler. CCCP inhibits the activation of STING and its downstream signaling molecules ...
T9137 SN-011 [1,1'-Biphenyl]-4-carboxamide, N-[3-[[(4-fluorophenyl)sulfonyl]amino]-4-hydroxyphenyl]-,GUN35901 STING
SN-011 (GUN35901) is a STING inhibitor, which inhibited the activation of the STING signal pathway and to prevent or treat a STING- mediated disease. It is a demethyl analogue of DUN99845.
T10252L2 ADU-S100 ammonium salt ML RR-S2 CDA ammonium salt,MIW815 ammonium salt STING
ADU-S100 ammonium salt (ML RR-S2 CDA ammonium salt) is an activator of stimulator of interferon genes (STING). ADU-S100 ammonium salt leads to potent and systemic tumor regression and immunity.
T6273 Vadimezan DMXAA,5,6-Dimethylxanthenone-4-acetic Acid,NSC 640488,ASA-404 Influenza Virus , VDA , STING , IFNAR
Vadimezan (DMXAA) is a vascular disrupting agent, a murine STING agonist, and an inducer of cytokines such as type I IFN. Vadimezan has antitumor activity and induces a rapid cessation of blood flow in tumors without aff...
T11035 DiABZI STING agonist-1 (Tautomerism) diABZI STING agonist (Compound 3) STING
diABZI STING agonist-1 (Tautomerism) (diABZI STING agonist (Compound 3)) is a selective stimulator of interferon genes (STING) receptor agonist, with EC50s of 130, 186 nM for human and mouse, respectively.
T68087 Inaperisone Others
Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.
T0511 Tolperisone hydrochloride Muscalm,Midocalm,Tolperisone HCl Sodium Channel
Tolperisone hydrochloride (Muscalm), a centrally acting muscle relaxant, is used in the therapy of pathologically increased tone of the cross-striated muscle resulted by neurological diseases (damage of the encephalomyel...
T5005 Eperisone hydrochloride Others
Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.
T8441 Lerisetron 5-HT Receptor
Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.
T70489 Enerisant HCl P450 , Histamine Receptor
Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins.
T28778 Silperisone HCl RGH5002,SILA336,RGH-5002,Silperisone hydrochloride,SILA-336
Silperisone HCl (RGH-5002) blocks sodium and calcium channels in cells, decreases excitability and contractility of muscle cells, reduces peripheral tone, and acts as a muscle relaxant and peripheral vasodilator. Silperi...
T28159 Nerisopam EGIS-6775,GYKI 52322,GYKI52322,EGIS6775,GYKI-52322 GABA Receptor
Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.
T32561 Lanperisone
Lanperisone is a muscle relaxant.
T28160 Nerispirdine HCl HP-184,HP 184,Nerispirdine hydrochloride,HP184
Nerispirdine is a acetylcholine release enhancer, sodium channel blocker and K(V) 2.1 channel blocker. Nerispirdine inhibits voltage-dependent Na(+) channel currents recorded from human SH-SY5Y cells with an IC(50) of 11...
T124126 Asteriscunolide A
Asteriscunolide A is a useful organic compound for research related to life sciences and the catalog number is T124126.
T40744 Eperisone
Eperisone is a centrally acting muscle relaxant and antispastic agent utilized in the treatment of conditions distinguished by muscle stiffness and pain. Its mechanism of action involves the relaxation of skeletal muscle...
T21077 Tolperisone free base Mydeton,Atmosgen free base,Mideton,Menopatol,Besnoline free base,Mydocalm
Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and muscle spasm.
T71356 Lanperisone HCl
Lanperisone, also known as NK433, is a muscle relaxant. NK433 inhibited the facilitation of the flexor reflex mediated by group II afferent fibers that was induced by intrathecal administration of noradrenaline-HCl. NK43...
T81509 Perisulfakinin
Perisulfakinin, a satiety-signaling neuropeptide, suppresses the activity of neurons that stimulate general activity [1].
T67828 Enerisant
Enerisant is an antagonist/inverse agonist of histamine H3 receptor.In vitro studies have shown that enerisant is a potent, highly selective, and competitive antagonist for the histamine H3 receptor, with a more than 3,0...
T125082 Pierisformoside B
Pierisformoside B is a useful organic compound for research related to life sciences. The catalog number is T125082 and the CAS number is 308335-44-6.
T125924 Pterisolic acid B
Pterisolic acid B is a useful organic compound for research related to life sciences and the catalog number is T125924.
T71281 Nerispirdine
Nerispirdine is a biochemical that inhibits batrachotoxin binding to voltage-dependent sodium channels.
T125921 Monnieriside A
Monnieriside A is a useful organic compound for research related to life sciences and the catalog number is T125921.

Compounds

STING agonist-4
T13015
Synonym:
Target: STING
ChX710
T13613
Synonym:
Target: STING
C-178
T7329
Synonym:
Target: STING
STING activator Compound 53
T9853
Synonym:
Target: STING
Omaveloxolone
T6919
Synonym: RTA-408
Target: Apoptosis, Others, Nrf2, STING
SN-008
T9554
Synonym:
Target: STING
H-151
T5674
Synonym:
Target: STING
SR-717
T8655
Synonym:
Target: STING
MSA-2
T8798
Synonym:
Target: STING
STING-IN-3
T9029
Synonym: C-171
Target: STING
C-176
T5154
Synonym: C176,STING inhibitor 1
Target: STING
diABZI STING agonist-1 trihydrochloride
T5516
Synonym:
Target: STING
STING agonist-1
T8328
Synonym: G10
Target: Virus Protease, STING
STING-IN-2
T9028
Synonym: C-170
Target: STING
CCCP
T7081
Synonym: Carbonyl Cyanide m-Chlorophenylhydrazone,Carbonyl cyanide 3-chlorophenylhydrazone
Target: Apoptosis, IκB/IKK, COX, Mitochondrial Metabolism, STING, IFNAR, Antibacterial
SN-011
T9137
Synonym: [1,1'-Biphenyl]-4-carboxamide, N-[3-[[(4-fluorophenyl)sulfonyl]amino]-4-hydroxyphenyl]-,GUN35901
Target: STING
ADU-S100 ammonium salt
T10252L2
Synonym: ML RR-S2 CDA ammonium salt,MIW815 ammonium salt
Target: STING
Vadimezan
T6273
Synonym: DMXAA,5,6-Dimethylxanthenone-4-acetic Acid,NSC 640488,ASA-404
Target: Influenza Virus, VDA, STING, IFNAR
diABZI STING agonist-1 (Tautomerism)
T11035
Synonym: diABZI STING agonist (Compound 3)
Target: STING
Inaperisone
T68087
Synonym:
Target: Others
Tolperisone hydrochloride
T0511
Synonym: Muscalm,Midocalm,Tolperisone HCl
Target: Sodium Channel
Eperisone hydrochloride
T5005
Synonym:
Target: Others
Lerisetron
T8441
Synonym:
Target: 5-HT Receptor
Enerisant HCl
T70489
Synonym:
Target: P450, Histamine Receptor
Silperisone HCl
T28778
Synonym: RGH5002,SILA336,RGH-5002,Silperisone hydrochloride,SILA-336
Target:
Nerisopam
T28159
Synonym: EGIS-6775,GYKI 52322,GYKI52322,EGIS6775,GYKI-52322
Target: GABA Receptor
Lanperisone
T32561
Synonym:
Target:
Nerispirdine HCl
T28160
Synonym: HP-184,HP 184,Nerispirdine hydrochloride,HP184
Target:
Asteriscunolide A
T124126
Synonym:
Target:
Eperisone
T40744
Synonym:
Target:
Tolperisone free base
T21077
Synonym: Mydeton,Atmosgen free base,Mideton,Menopatol,Besnoline free base,Mydocalm
Target:
Lanperisone HCl
T71356
Synonym:
Target:
Perisulfakinin
T81509
Synonym:
Target:
Enerisant
T67828
Synonym:
Target:
Pierisformoside B
T125082
Synonym:
Target:
Pterisolic acid B
T125924
Synonym:
Target:
Nerispirdine
T71281
Synonym:
Target:
Monnieriside A
T125921
Synonym:
Target:
Cat No. Product Name Synonyms Targets
TN4843 Pterisolic acid A Others
Pterisolic acid A shows moderate activity against HCT-116,Hep G2 and BGC-823 cell lines.
T81766 Monnierisides A
Monnierisides A, a chromone glycoside, has been isolated from Cnidium monnieri [1].
TN2056 Perisesaccharide B Others
Perisesaccharide B is a natural product
TN1356 Acetyl Perisesaccharide C Others
Acetyl Perisesaccharide C is a natural product
TN4846 Pterisolic acid F Others
Pterisolic acid F is a natural product from Pteris semipinnata.
TN1948 Monnieriside G Others
Monnieriside G is a natural product from Cnidium monnieri.
TN5576 Pterisolic acid E
Pterisolic acid E is a natural product from Pteris semipinnata.
TN4845 Pterisolic acid D Others
Pterisolic acid D is a natural product for research related to life sciences. The catalog number is TN4845 and the CAS number is 1401419-88-2.
TN2057 Perisesaccharide C Others
Perisesaccharide C is a natural product
T83260 6β,7β-Epoxyasteriscunolide A
6β,7β-Epoxyasteriscunolide A, a sesquiterpenoid, exhibits cytotoxicity against HL-60 and MOLT-3 leukemia cell lines, demonstrating half maximal inhibitory concentrations (IC50s) ranging from 4.1 to 5.4 μM [1].
TN4844 Pterisolic acid C Others
Pterisolic acid C is a natural product from Pteris semipinnata.

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPH-00363 Cyanovirin-N homolog Protein, Ceratopteris richardii, Recombinant (His) Ceratopteris richardii Yeast
Mannose-binding lectin.
TargetMol