T12911 |
Sigma-1 receptor antagonist 2
|
1639220-15-7
|
98%
|
|
Sigma-1 receptor antagonist 2 is a potent and selective antagonist of sigma 1 receptor (σ1 R) (σ1 and σ2 receptor with Kis of 3.88 and 1288 nM , respectively).
|
T3198L |
PRE-084 hydrochloride
|
75136-54-8
|
98%
|
|
PRE-084 hydrochloride is a selective agonist of σ1(IC50:44 nM, in the sigma receptor assay).
|
T22240 |
Amitriptyline
|
50-48-6
|
98%
|
|
Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties. Amitriptyline is widely used to treat depression and neurop...
|
T9244 |
σ1 Receptor antagonist-1
|
1204401-49-9
|
98%
|
|
σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.
|
T1885 |
Siramesine hydrochloride
|
224177-60-0
|
98%
|
|
Siramesine (Lu 28-179) hydrochloride is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit a potent antic...
|
T15393 |
Glycerol phenylbutyrate
|
611168-24-2
|
98%
|
|
Glycerol phenylbutyrate (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).
|
T4229 |
S1RA hydrochloride
|
1265917-14-3
|
98%
|
|
S1RA HCl (E-52862 HCl) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki > 1000 nM).
|
T12910 |
Sigma-1 receptor antagonist 1
|
1639220-19-1
|
98%
|
|
Sigma-1 receptor antagonist 1 is an effective and selective antagonist of sigma-1 receptor. Sigma-1 receptor antagonist 1 exhibits antineuropathic pain activity ...
|
T0678 |
Amitriptyline hydrochloride
|
549-18-8
|
98%
|
|
Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.
|
T5027 |
Dimemorfan phosphate
|
36304-84-4
|
98%
|
|
Dimemorfan phosphate is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.
|
T4111 |
Blarcamesine hydrochloride
|
195615-84-0
|
98%
|
|
Anavex 2-73 is a Sigma-1 Receptor agonist (IC50: 860 nM).
|
T3597 |
Cutamesine dihydrochloride
|
165377-44-6
|
98%
|
|
Cutamesine dihydrochloride is a selective σ1 receptor agonist (IC50: 17.4 nM). It shows selectivity for σ1 over σ2 receptors, and inhibits angiotensin II-induced...
|
T3198 |
Pre-084
|
138847-85-5
|
98%
|
|
PRE-084 hydrochloride is a high affinity, selective σ1 agonist.
|