T23077L |
Novokinin acetate
|
T23077L
|
98%
|
|
Novokinin acetate exhibited an affinity for the AT2 receptor with Ki of 7 nM, and its antihypertensive and vasorelaxing activities were blocked by PD123319, an A...
|
T35834L |
(Sar¹)-Angiotensin II acetate
|
T35834L
|
98%
|
|
(Sar¹)-Angiotensin II acetate, an analogue of Angiotensin II, is a specific agonist of angiotensin AT1 receptor. It binds to brain membrane-rich particles, with ...
|
T3064 |
VTP-27999
|
942142-51-0
|
98%
|
|
VTP-27999 is an alkyl amine Renin inhibitor. VTP-27999 has been used in trials studying the basic science of Renal Function.
|
T3178 |
BIBS 39
|
133085-33-3
|
98%
|
|
BIBS 39 is a new nonpeptide angiotensin II (AII) receptor antagonist.
|
T7743 |
ANGIOTENSIN IV TFA(12676-15-2(free base))
|
T7743
|
98%
|
|
ANGIOTENSIN IV TFA is a less effective agonist at the angiotensin AT1 receptor.
|
T7577 |
Angiotensin III, human, mouse
|
13602-53-4
|
98%
|
|
Angiotensin III, human, mouse(3TFA) is an endogenous angiotensin II receptor (AT2R) agonist(IC50s of 0.648 nM).
|
T7354 |
H-Val-Pro-Pro-OH
|
58872-39-2
|
98%
|
|
H-Val-Pro-Pro-OH is an inhibitor of Angiotensin I converting enzyme (ACE)( IC50 : 9 μM).
|
TP1528 |
Angiotensin I/II (1-5)
|
58442-64-1
|
98%
|
|
Angiotensin I/II (1-5) is a peptide (ASP-ARG-VAL-TYR-ILE) that contains the amino acids 1-5 and is converted from Angiotensin I/II.
|
T2400 |
Candesartan Cilexetil
|
145040-37-5
|
98%
|
|
Candesartan Cilexetil is an angiotensin II receptor antagonist (IC50: 0.26 nM). After hydrolysis of candesartan cilexetil to candesartan during gastrointestinal ...
|
TP1016L |
Aviptadil Acetate
|
1444827-29-5
|
98%
|
|
Avitadil acetate induces pulmonary vasodilation and inhibits the proliferation of vascular SMCs and platelet aggregation. Avitadil acetate can be used for resear...
|
T7616L |
A 779 TFA(159432-28-7 free base)
|
T7616L
|
98%
|
|
A 779(3TFA) is a potent antagonist of angiotensin-(1-7) receptor
|
T7510 |
Leucylarginylproline
|
133943-59-6
|
98%
|
|
Leucylarginylproline is an inhibitor of angiotensin-converting enzyme (ACE) (IC50 : 0.27μM).
|
T7339 |
Angiotensin (1-7)
|
51833-78-4
|
98%
|
|
Angiotensin 1-7, also known as Ang-(1-7), is a synthetic heptapeptide identical to endogenous angiotensin-(1-7) , inhibits purified canine ACE activity (IC50=0.6...
|
T0215 |
Losartan potassium
|
124750-99-8
|
98%
|
|
Losartan, an Angiotensin II Receptor Blocker, selectively and competitively blocks the binding of angiotensin II to the angiotensin I (AT1) receptor.
|
T6595 |
Moexipril hydrochloride
|
82586-52-5
|
98%
|
|
Moexipril HCl is a potent orally active nonsulfhydrylangiotensin converting enzyme (ACE)inhibitor, used for the treatment of hypertension and congestive heart fa...
|
T4431 |
Olodanrigan
|
1316755-16-4
|
98%
|
|
EMA401, a highly selective AT2R antagonist, inhibition of augmented AngII/AT2R induced p38 and p42/p44 MAPK activation, and hence inhibition of DRG neuron hypere...
|
TP2158 |
TRV-120027 TFA
|
TP2158
|
98%
|
|
TRV120027 TFA is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1R) and engages ß-arrestins while blocking G-protein signaling.
|
T14337 |
Buloxibutid
|
477775-14-7
|
98%
|
|
Buloxibutid is a novel and selective small molecule angiotensin II AT2 receptor agonist with Ki values of 0.4 nM and 10 μM for AT2 and AT1 receptors, respectivel...
|
T6219 |
Azilsartan Medoxomil
|
863031-21-4
|
98%
|
|
Azilsartan medoxomil(TAK 491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults wit...
|
T2322 |
Fimasartan
|
247257-48-3
|
98%
|
|
Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Concurrent administration of fimas...
|