T15368L |
Galantide acetate
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97.8%
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Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two ...
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T23094 |
NTNCB hydrochloride
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191931-56-3
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97.92%
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NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
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TP1074L |
Neuropeptide FF acetate(99566-27-5 free base)
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TP1074L
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98.03%
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NPFF acetate is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).
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TP1884L1 |
Neuropeptide SF(mouse,rat) acetate
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TP1884L1
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98.37%
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Neuropeptide SF (mouse,rat) acetate is a potent neuropeptide FF receptor agonist, Ki for NPFF1 and NPFF2 are 48.4 nM and 12.1 nM, respectively. Neuropeptide SF (...
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T5455 |
HT-2157
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303149-14-6
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98.55%
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HT-2157 is a selective, high-affinity, competitive antagonists of galanin-3 receptor (Gal3).
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T10539 |
BIBO3304 TFA
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191868-14-1
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98.87%
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BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recept...
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T23087 |
NPY 5RA972
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439861-56-0
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99.02%
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neuropeptide Y Y5 receptor antagonist
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TP1991L |
M 1145 acetate
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99.1%
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M1145 acetate, a chimeric peptide, is a selective galanin receptor type 2 (GAL2) agonist, with a Ki of 6.55 nM. M1145 acetate shows more than 90-fold higher affi...
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T16738L |
RF9 acetate
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99.35%
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RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
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T22994 |
ML 154
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1345964-89-7
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99.44%
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neuropeptide S receptor (NPSR) antagonist
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TP1704 |
Galanin Receptor Ligand M35 TFA
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TP1704
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99.45%
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Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).
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TQ0286 |
MK-0557
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328232-95-7
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99.81%
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MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
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T5587 |
CGP71683 hydrochloride
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192322-50-2
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99.82%
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CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM...
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T17222 |
Velneperit
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342577-38-2
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99.82%
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Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
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TP1992L |
M40 acetate(143896-17-7 free base)
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TP1992L
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99.88%
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M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) bi...
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T8559 |
GALNON TFA(475115-35-6(free base))
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T8559
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99.92%
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Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).
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T22608 |
BMS 193885
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679839-66-8
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98%
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BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.
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T21611L |
BWX 46 Acetate
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T21611L
|
98%
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BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
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TP1930L1 |
Spexin acetate(1370290-58-6 free base)
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TP1930L1
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98%
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Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galani...
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