T22994 |
ML 154
|
1345964-89-7
|
99.44%
|
|
neuropeptide S receptor (NPSR) antagonist
|
T16738L |
RF9 acetate
|
|
99.35%
|
|
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
|
TP1991L |
M 1145 acetate
|
|
99.1%
|
|
M1145 acetate, a chimeric peptide, is a selective galanin receptor type 2 (GAL2) agonist, with a Ki of 6.55 nM. M1145 acetate shows more than 90-fold higher affi...
|
T23087 |
NPY 5RA972
|
439861-56-0
|
99.02%
|
|
neuropeptide Y Y5 receptor antagonist
|
T10539 |
BIBO3304 TFA
|
191868-14-1
|
98.87%
|
|
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recept...
|
T5455 |
HT-2157
|
303149-14-6
|
98.55%
|
|
HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.
|
TP1884L1 |
Neuropeptide SF(mouse,rat) acetate
|
TP1884L1
|
98.37%
|
|
Neuropeptide SF(mouse,rat) acetate (Neuropeptide SF(mouse,rat) acetate (230960-31-3 free base)) is a potent neuropeptide FF receptor agonist, Ki for NPFF1 and NP...
|
TP1074L |
Neuropeptide FF acetate(99566-27-5 free base)
|
TP1074L
|
98.03%
|
|
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors ...
|
T23094 |
NTNCB hydrochloride
|
191931-56-3
|
97.92%
|
|
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
|
T15368L |
Galantide acetate
|
|
97.8%
|
|
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two ...
|
TP1936L1 |
RFRP3(human) acetate(311309-27-0 free base)
|
TP1936L1
|
97.09%
|
|
RFRP-3(human) acetate, a human GnIH peptide homolog, is a potent inhibitor of gonadotropin secretion by inhibiting Ca2+ mobilization. RFRP-3(human) acetate is a ...
|
T8963 |
CYM2503
|
1308833-36-4
|
97.04%
|
|
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthos...
|
T21611L |
BWX 46 Acetate
|
T21611L
|
96.86%
|
|
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
|
TP1937L1 |
RFRP-1 (human) acetate(311309-25-8 free base)
|
TP1937L1
|
96.84%
|
|
RFRP-1 (human) acetate is a potent endogenous NPFF receptor agonist (EC50 values are 0.0011 and 29 nM for NPFF2 and NPFF1, respectively). Attenuates contractile ...
|
TP1930L1 |
Spexin acetate(1370290-58-6 free base)
|
TP1930L1
|
95.43%
|
|
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galani...
|
T21646L |
AR-M 1896 Acetate
|
T21646L
|
95.32%
|
|
AR-M 1896 Acetate is the selective agonist of GalR2.
|
T24121 |
GW438014A
|
469861-49-2
|
100%
|
|
GW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and curbing body weight gain in obese rodents.
|
T10056 |
Neurokinin antagonist 1
|
214487-45-3
|
100%
|
|
Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.
|
T1997 |
JNJ-31020028
|
1094873-14-9
|
|
|
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold ...
|
T71749 |
SF-22
|
824981-55-7
|
98%
|
|
SF-22 is a neuropeptide Y receptor (Y2R) antagonist that crosses the blood-brain barrier and has potential anti-inflammatory activity for the study of diseases a...
|