Neuropeptide Y Receptor

Neuropeptide Y receptors are a family of receptors belonging to class A G-protein coupled receptors and they are activated by the closely related peptide hormones neuropeptide Y, peptide YY and pancreatic polypeptide. These receptors are involved in the control of a diverse set of behavioral processes including appetite, circadian rhythm, and anxiety.

Cat. No.	Product name	CAS No.	Purity
T15368L	Galantide acetate		97.8%
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two ...
T23094	NTNCB hydrochloride	191931-56-3	97.92%
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
TP1074L	Neuropeptide FF acetate(99566-27-5 free base)	TP1074L	98.03%
NPFF acetate is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).
TP1884L1	Neuropeptide SF(mouse,rat) acetate	TP1884L1	98.37%
Neuropeptide SF (mouse,rat) acetate is a potent neuropeptide FF receptor agonist, Ki for NPFF1 and NPFF2 are 48.4 nM and 12.1 nM, respectively. Neuropeptide SF (...
T5455	HT-2157	303149-14-6	98.55%
HT-2157 is a selective, high-affinity, competitive antagonists of galanin-3 receptor (Gal3).
T10539	BIBO3304 TFA	191868-14-1	98.87%
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recept...
T23087	NPY 5RA972	439861-56-0	99.02%
neuropeptide Y Y5 receptor antagonist
TP1991L	M 1145 acetate		99.1%
M1145 acetate, a chimeric peptide, is a selective galanin receptor type 2 (GAL2) agonist, with a Ki of 6.55 nM. M1145 acetate shows more than 90-fold higher affi...
T16738L	RF9 acetate		99.35%
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
T22994	ML 154	1345964-89-7	99.44%
neuropeptide S receptor (NPSR) antagonist
TP1704	Galanin Receptor Ligand M35 TFA	TP1704	99.45%
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).
TQ0286	MK-0557	328232-95-7	99.81%
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
T5587	CGP71683 hydrochloride	192322-50-2	99.82%
CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM...
T17222	Velneperit	342577-38-2	99.82%
Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
TP1992L	M40 acetate(143896-17-7 free base)	TP1992L	99.88%
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) bi...
T8559	GALNON TFA(475115-35-6(free base))	T8559	99.92%
Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).
T22608	BMS 193885	679839-66-8	98%
BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.
T21611L	BWX 46 Acetate	T21611L	98%
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
TP1930L1	Spexin acetate(1370290-58-6 free base)	TP1930L1	98%
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galani...

Cat. No.

Product name

CAS No.

Purity

Chemical Structure

T15368L

Galantide acetate

97.8%

Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two ...

T23094

NTNCB hydrochloride

191931-56-3

97.92%

NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.

TP1074L

Neuropeptide FF acetate(99566-27-5 free base)

TP1074L

98.03%

NPFF acetate is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).

TP1884L1

Neuropeptide SF(mouse,rat) acetate

TP1884L1

98.37%

Neuropeptide SF (mouse,rat) acetate is a potent neuropeptide FF receptor agonist, Ki for NPFF1 and NPFF2 are 48.4 nM and 12.1 nM, respectively. Neuropeptide SF (...

T5455

HT-2157

303149-14-6

98.55%

HT-2157 is a selective, high-affinity, competitive antagonists of galanin-3 receptor (Gal3).

T10539

BIBO3304 TFA

191868-14-1

98.87%

BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recept...

T23087

NPY 5RA972

439861-56-0

99.02%

neuropeptide Y Y5 receptor antagonist

TP1991L

M 1145 acetate

99.1%

M1145 acetate, a chimeric peptide, is a selective galanin receptor type 2 (GAL2) agonist, with a Ki of 6.55 nM. M1145 acetate shows more than 90-fold higher affi...

T16738L

RF9 acetate

99.35%

RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.

T22994

ML 154

1345964-89-7

99.44%

neuropeptide S receptor (NPSR) antagonist

TP1704

Galanin Receptor Ligand M35 TFA

TP1704

99.45%

Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).

TQ0286

MK-0557

328232-95-7

99.81%

MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).

T5587

CGP71683 hydrochloride

192322-50-2

99.82%

CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM...

T17222

Velneperit

342577-38-2

99.82%

Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.

TP1992L

M40 acetate(143896-17-7 free base)

TP1992L

99.88%

M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) bi...

T8559

GALNON TFA(475115-35-6(free base))

T8559

99.92%

Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).

T22608

BMS 193885

679839-66-8

98%

BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.

T21611L

BWX 46 Acetate

T21611L

98%

BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.

TP1930L1

Spexin acetate(1370290-58-6 free base)

TP1930L1

98%

Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galani...