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Melanocortin Receptor

Melanocortin receptors are members of the rhodopsin family of 7-transmembrane G protein-coupled receptors. There are five known members of the melanocortin receptor system:MC1R,MC2R,MC3R,MC4R,MC5R.
Cat. No. Product name CAS No. Purity Chemical Structure
T12882 Setmelanotide 920014-72-8 98%
Setmelanotide is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
T7627 Adrenocorticotropic Hormone (ACTH) (4-10), human 4037-01-8 98%
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
T20501 Undecylenoyl phenylalanine 175357-18-3 98%
Undecylenoyl phenylalanine is a novel, skin-lightening agent. It acting as α-melanocyte-stimulating hormone and beta-adrenergic receptor antagonist.
T16879L SHU 9119 acetate T16879L
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
TP1898 HS024 212370-59-7 100%
Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). In...
T7813 α-MSH 581-05-5 100%
α-MSH is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
TP1893L1 [D-Trp8]-γ-MSH acetate(321351-81-9 free base) TP1893L1 100%
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
TP1324 Melanotan (MT)-II 121062-08-6 100%
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
TP1248L ACTH 11-24 acetate(4237-93-8 free base) TP1248L 100%
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
T12882L Setmelanotide Acetate(920014-72-8 free base) T12882L 100%
Setmelanotide Acetate is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
TP2015L HS 014 acetate(207678-81-7 free base) TP2015L 100%
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 re...
T7608 Bremelanotide Acetate 1607799-13-2 98%
Bremelanotide is an agonist of melanocortin receptor (MCR) .
T7589 Afamelanotide acetate 1566590-77-9 98%
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
TP1101 Nonapeptide-1 acetate salt (158563-45-2 free base) TP1101 98%
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
TP1952L PG 106 acetate 98.24%
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
TP2212L A-MSH, amide Acetate(581-05-5 free base) TP2212L 98.67%
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
T8485 THIQ 312637-48-2 98.93%
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
T7627L Adrenocorticotropic Hormone (ACTH) (4-10) TFA T7627L 99%
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
T5464 JNJ-10229570 524923-88-4 99.06%
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
TP1889 MCL0020 475498-26-1 99.18%
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
Setmelanotide
T12882
Setmelanotide is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
Adrenocorticotropic Hormone (ACTH) (4-10), human
T7627
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
Undecylenoyl phenylalanine
T20501
Undecylenoyl phenylalanine is a novel, skin-lightening agent. It acting as α-melanocyte-stimulating hormone and beta-adrenergic receptor antagonist.
SHU 9119 acetate
T16879L
SHU 9119 acetate is a well-known antagonist of human melanocortin 3 and 4 (hMC3R, hMC4R) receptors and a partial hMC5R agonist. The IC50 values of human MC3R, MC...
HS024
TP1898
Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). In...
α-MSH
T7813
α-MSH is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.
[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
TP1893L1
Selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively). Displays anti-inflammato...
Melanotan (MT)-II
TP1324
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
ACTH 11-24 acetate(4237-93-8 free base)
TP1248L
ACTH (11-24) acetate is a fragment of adrenocorticotrophin, induces cortisol release. ACTH (11-24) has been identified as a competitive antagonist of ACTH (1-39)...
Setmelanotide Acetate(920014-72-8 free base)
T12882L
Setmelanotide Acetate is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).
HS 014 acetate(207678-81-7 free base)
TP2015L
HS 014 acetate is a potent and selective melanocortin MC4 receptor antagonist (Ki values are 3.16, 108, 54.4 and 694 nM for cloned human MC4, MC1, MC3 and MC5 re...
Bremelanotide Acetate
T7608
Bremelanotide is an agonist of melanocortin receptor (MCR) .
Afamelanotide acetate
T7589
Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist, used to for Erythropoietic Pro...
Nonapeptide-1 acetate salt (158563-45-2 free base)
TP1101
Nonapeptide-1 acetate salt, a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH) antagonist, with an IC50 of 11 nM. Nonapeptide-1 acetate salt...
PG 106 acetate
TP1952L
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with t...
a-MSH, amide Acetate(581-05-5 free base)
TP2212L
a-MSH, amide Acetate as an endogenous neuropeptide. It is an endogenous melanocortin receptor 4 (MC4R) agonist with anti-inflammatory and antipyretic activities....
THIQ
T8485
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).
Adrenocorticotropic Hormone (ACTH) (4-10) TFA
T7627L
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
JNJ-10229570
T5464
JNJ-10229570 is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland differentiation and the produc...
MCL0020
TP1889
Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly...
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