Cat. No. | Product name | CAS No. | Purity | Chemical Structure |
---|---|---|---|---|
T5428 | BIX 02565 | 1311367-27-7 | 98% |
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BIX 02565 is a potent inhibitor of ribosomal S6 kinase 2 (RSK2, IC50: 1.1 nM). | ||||
T39972 | EB-42486 | 2390475-81-5 | 98% |
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EB-42486 is an effective and highly selective inhibitor of G2019S-LRRK2 with an IC50 < 0.2 nM. | ||||
T6057 | URMC-099 | 1229582-33-5 | 98% |
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URMC-099 is an orally bioavailable, brain penetrant MLK inhibitor (IC50: 19/42/14/150 nM, for MLK1/MLK2/MLK3/DLK), and also inhibits LRRK2 activity (IC50: 11 nM)... |