GluR

Glutamate receptors are synaptic and non synaptic receptors located primarily on the membranes of neuronal and glial cells.Glutamate receptors are responsible for the glutamate-mediated postsynaptic excitation of neural cells, and are important for neural communication, memory formation, learning, and regulation.

Cat. No.	Product name	CAS No.	Purity
T3464	PHCCC	179068-02-1	99.31%
T3464	PHCCC is a Group I metabotropic glutamate receptor antagonist and a positive allosteric modulator of mGluR4. It also is a potent to antagonism for mGluR2 and mGl...
T0326L	L-Glutamine	56-85-9	99.36%
T0326L	L-glutamine, a non-essential amino acid, is synthesized from glutamic acid and ammonia.
T12717	Basimglurant	802906-73-6	99.38%
T12717	Basimglurant is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd of 1.1 nM).
T15090	Decoglurant	911115-16-7	99.39%
T15090	Decoglurant is a negative allosteric modulator of mGluR2 and mGluR3 and it also is developed as an antidepressant.
T22641	CDPPB	781652-57-1	99.39%
T22641	CDPPB is a modulator of mGluR5 positive allosteric(with an EC50 of 27 nM in Chinese hamster ovary cells expressing human mGluR5).
T5512	JNJ16259685	409345-29-5	99.39%
T5512	JNJ16259685 is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19 nM.
T3473	(S)-ATPO	252930-37-3	99.41%
T3473	ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.
TP2111L	TAT-GluA2 3Y acetate(1404188-93-7 free base)	TP2111L	99.43%
TP2111L	TAT-GluA2 3Y acetate is an inhibitor of AMPA receptor endocytosis. Induces increased hind paw withdrawal latencies following thermal and mechanical stimuli in ra...
T15275	Fenobam	57653-26-6	99.44%
T15275	Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM). Fenobam has anxiolytic activity. Fenobam is a selective and n...
T2811	Harmine hydrochloride	343-27-1	99.45%
T2811	Harmine hydrochloride is extracted from Peganum Harmala Genus.
T6871	L-Glutamic acid monosodium salt	142-47-2	99.45%
T6871	L-Glutamic acid monosodium salt (Monosodium glutamate) is an activator of mGlu1 receptor.
T23515	VU-29	890764-36-0	99.47%
T23515	VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes (EC...
T3478	Ro 67-7476	298690-60-5	99.48%
T3478	Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors. No activity at human mGlu1 receptors. Potentiates glutamate-induced calcium release with EC 50 ...
T8779	HBT1	489408-02-8	99.48%
T8779	HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons....
T8626	4-oxo-1,4-dihydroquinoline-2-carboxylic acid	13593-94-7	99.49%
T8626	4-oxo-1,4-dihydroquinoline-2-carboxylic acid is a GluR and NMDA inhibitor.
T10432L	AZD-8529 mesylate	1314217-69-0	99.5%
T10432L	AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM). It shows no positive allosteric modulato...
T3484	Trans-ACPD	67684-64-4	99.53%
T3484	(±)-trans-ACPD is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD. (±)-trans-ACPD is a selective agonist of the mGluR (metabotropic glutamate receptor); ...
T11393	GET73	202402-01-5	99.54%
T11393	GET73 is an negative allosteric modulator of mGluR5. GET73 is a naturally occurring neurotransmitter. GET73 has anti-alcohol and anxiolytic properties.
T11032	DHPG	146255-66-5	99.55%
T11032	DHPG ((RS)-3,5-DHPG) is an effective antagonist of mGluR linked to phospholipase D. It is an amino acid that can be used as a selective and potent agonist for Gr...
T3565	VU0155041	1093757-42-6	99.56%
T3565	UV0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).