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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Cat. No. Product name CAS No. Purity Chemical Structure
T3403 Glabridin 59870-68-7 98%
Glabridin may serve as an anti-inflammatory agent in diabetes-related vascular dysfunction, through regulating the synthesis and activity of iNOS under high-gluc...
T1065 Baclofen 1134-47-0 98%
Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing Baclofen act...
T8036 6-Methylflavone 29976-75-8 98%
6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
T4590 (+)-Kavain 500-64-1 98%
Kawain is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.
T26891 BPDBA 312281-74-6 98%
T7699 AZD7325 942437-37-8 98%
AZD-7325 is a GABA-Aα2,3 -selective receptor modulator.
T0349 Riluzole 1744-22-5 98%
Riluzole is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LA...
T5330 Fluralaner 864731-61-3 98%
Fluralaner is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head membranes ...
T1240 Flumazenil 78755-81-4 98%
Flumazenil antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous system (CNS),...
T0710 L-Cycloserine 339-72-0 98%
L-cycloserine irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminotransferase in E. coli, as well in the brains of various animals, results in incre...
T13536 Afoxolaner 1093861-60-9 98%
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA...
T8639 Phenibut (hydrochloride) 3060-41-1 98%
Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates d...
T5375 Loreclezole 117857-45-1 98%
Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
T2S1464 Thiocolchicoside 602-41-5 98%
Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonis...
T3644 U93631 152273-12-6 98%
GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GAB...
T0715 Chlormezanone 80-77-3 98%
Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
T2339 Apalutamide 956104-40-8 98%
Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T8572 CL 218872 66548-69-4 98%
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 n...
T1396 Bemegride 64-65-3 98%
Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning.
T2850 Bicuculline 485-49-4 98%
Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated...
Glabridin
T3403
Glabridin may serve as an anti-inflammatory agent in diabetes-related vascular dysfunction, through regulating the synthesis and activity of iNOS under high-gluc...
Baclofen
T1065
Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing Baclofen act...
6-Methylflavone
T8036
6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
(+)-Kavain
T4590
Kawain is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.
BPDBA
T26891
AZD7325
T7699
AZD-7325 is a GABA-Aα2,3 -selective receptor modulator.
Riluzole
T0349
Riluzole is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LA...
Fluralaner
T5330
Fluralaner is an isoxazoline ectoparasiticide. It potently and selectively inhibits binding of the GABA receptor channel blocker EBOB to housefly head membranes ...
Flumazenil
T1240
Flumazenil antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous system (CNS),...
L-Cycloserine
T0710
L-cycloserine irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminotransferase in E. coli, as well in the brains of various animals, results in incre...
Afoxolaner
T13536
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA...
Phenibut (hydrochloride)
T8639
Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates d...
Loreclezole
T5375
Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
Thiocolchicoside
T2S1464
Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonis...
U93631
T3644
GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GAB...
Chlormezanone
T0715
Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
Apalutamide
T2339
Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
CL 218872
T8572
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 n...
Bemegride
T1396
Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning.
Bicuculline
T2850
Bicuculline is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and has been isolated...
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