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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Cat. No. Product name CAS No. Purity Chemical Structure
T17144 TPA 023 252977-51-8 98%
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).
T23039 N-Arachidonyl-GABA 128201-89-8 98%
N-Arachidonyl-GABA (NA-GABA) is a novel active fatty amino acid related to anandamide (ANA) found in cattle. NA-GABA has analgesic activity
T0627 β-Alanine 107-95-9 98%
β-Alanine is a naturally occurring beta amino acid formed in vivo by the degradation of dihydrouracil and carnosine. It acts as a neurotransmitter by activating ...
T0883 Tramiprosate 3687-18-1 98%
Because of its similarity in structure to the neurotransmitter gamma-aminobutyric acid (GABA), it has GABAergic effects and may be useful as an anticonvulsant. H...
T1602 Valproic acid sodium salt 1069-66-5 98%
Valproate Sodium is the sodium salt form of valproic acid with anti-epileptic activity. Valproate sodium is converted into its active form, valproate ion, in blo...
T7557 Guvacine hydrochloride 6027-91-4 98%
Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
T10618 Broflanilide 1207727-04-5 98%
Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL ...
T38205 3-Aminopropylphosphonic Acid 13138-33-5 98%
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding as...
T23339 SCS 3232-36-8 98%
GABAA receptor antagonist
T11277 FG 7142 78538-74-6 98%
FG 7142 also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 can increase tyrosine hydroxylation and ca...
T22301 L-838417 D9 1213669-91-0 98%
L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].
T23104 Ocinaplon 96604-21-6 98%
GABAA receptors modulator
TN1217 2'-O-Methylisoliquiritigenin 51828-10-5 98%
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
T12930 SKF89976A hydrochloride 85375-15-1 98%
SKF89976A hydrochloride is a selective inhibitor of GABA transporter (GAT-1)(IC50s of 0.28 μM, 137.34 μM and 202.8 μM for GAT-1, GAT-2 and GAT-3 in CHO cells, re...
T15212 Emamectin Benzoate 155569-91-8 98%
Emamectin Benzoate, by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods, acts as ...
T3318 Wogonoside 51059-44-0 98%
Wogonoside acts as a positive allosteric modulator of the benzodiazepine site of the GABAA receptor.
T11822 LAU159 2055050-87-6 98%
LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
T7794 Zuranolone 1632051-40-1 98%
Zuranolone is an agonist of GABAA receptor.
T2775 Baicalin 21967-41-9 98%
Baicalin is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV properties.
T1860 Imepitoin 188116-07-6 98%
AWD 131-138(Imepitoin) is a new low-affinity partial benzodiazepine receptor agonist. It shows potent anticonvulsant and anxiolytic properties in rodent models.
TPA 023
T17144
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).
N-Arachidonyl-GABA
T23039
N-Arachidonyl-GABA (NA-GABA) is a novel active fatty amino acid related to anandamide (ANA) found in cattle. NA-GABA has analgesic activity
β-Alanine
T0627
β-Alanine is a naturally occurring beta amino acid formed in vivo by the degradation of dihydrouracil and carnosine. It acts as a neurotransmitter by activating ...
Tramiprosate
T0883
Because of its similarity in structure to the neurotransmitter gamma-aminobutyric acid (GABA), it has GABAergic effects and may be useful as an anticonvulsant. H...
Valproic acid sodium salt
T1602
Valproate Sodium is the sodium salt form of valproic acid with anti-epileptic activity. Valproate sodium is converted into its active form, valproate ion, in blo...
Guvacine hydrochloride
T7557
Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
Broflanilide
T10618
Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL ...
3-Aminopropylphosphonic Acid
T38205
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding as...
SCS
T23339
GABAA receptor antagonist
FG 7142
T11277
FG 7142 also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 can increase tyrosine hydroxylation and ca...
L-838417 D9
T22301
L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].
Ocinaplon
T23104
GABAA receptors modulator
2'-O-Methylisoliquiritigenin
TN1217
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
SKF89976A hydrochloride
T12930
SKF89976A hydrochloride is a selective inhibitor of GABA transporter (GAT-1)(IC50s of 0.28 μM, 137.34 μM and 202.8 μM for GAT-1, GAT-2 and GAT-3 in CHO cells, re...
Emamectin Benzoate
T15212
Emamectin Benzoate, by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods, acts as ...
Wogonoside
T3318
Wogonoside acts as a positive allosteric modulator of the benzodiazepine site of the GABAA receptor.
LAU159
T11822
LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
Zuranolone
T7794
Zuranolone is an agonist of GABAA receptor.
Baicalin
T2775
Baicalin is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV properties.
Imepitoin
T1860
AWD 131-138(Imepitoin) is a new low-affinity partial benzodiazepine receptor agonist. It shows potent anticonvulsant and anxiolytic properties in rodent models.
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