T13690 |
Etifoxine hydrochloride
|
56776-32-0
|
99.25%
|
|
Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug. Unlike benzodiazepines, Etifoxine hydrochloride appears to produce i...
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T26891 |
BPDBA
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312281-74-6
|
99.24%
|
|
BPDBA is a useful organic compound for research related to life sciences. The catalog number is T26891 and the CAS number is 312281-74-6.
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T2407 |
Tiagabine
|
115103-54-3
|
99.24%
|
|
Tiagabine (NO050328) is an Anti-epileptic Agent. The physiologic effect of tiagabine is by means of Decreased Central Nervous System Disorganized Electrical Acti...
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T2983 |
3,4,5-Trimethoxycinnamic acid
|
90-50-6
|
99.19%
|
|
3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the GA...
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T4363 |
CGP52432
|
139667-74-6
|
99.16%
|
|
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
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T3S2100 |
(-)-Securinine
|
5610-40-2
|
99.12%
|
|
(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.
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T77568 |
6,7-dimethylisatin
|
20205-43-0
|
99.09%
|
|
6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.
|
T23470 |
Tracazolate hydrochloride
|
1135210-68-2
|
99.07%
|
|
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity. Tracazolate hydrochlori...
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T17144 |
TPA 023
|
252977-51-8
|
99.06%
|
|
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).
|
T0627 |
β-Alanine
|
107-95-9
|
99%
|
|
β-Alanine (3-Aminopropanoic acid) is a naturally occurring beta amino acid formed in vivo by the degradation of dihydrouracil and carnosine. It acts as a neurotr...
|
T0883 |
Tramiprosate
|
3687-18-1
|
99%
|
|
Tramiprosate (Alzhemed) is an orally active, blood-brain-barrier-crossing, naturally occurring amino acid found in a variety of red seaweeds that binds soluble A...
|
T1602 |
Valproic acid sodium salt
|
1069-66-5
|
99%
|
|
Valproic acid sodium salt (Sodium Valproate) is the sodium salt form of valproic acid with anti-epileptic activity. Valproic acid sodium salt is converted into i...
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T2775 |
Baicalin
|
21967-41-9
|
98.96%
|
|
Baicalin (Baicalein 7-O-β-D-glucuronide) is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV proper...
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T7557 |
Guvacine hydrochloride
|
6027-91-4
|
98.96%
|
|
Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
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T10618 |
Broflanilide
|
1207727-04-5
|
98.95%
|
|
Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL ...
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T11061 |
DMCM hydrochloride
|
1215833-62-7
|
98.95%
|
|
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine. DMCM showed significant differences in human recombinant GABAA αxβ3γ2 receptor sub...
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T38205 |
3-Aminopropylphosphonic Acid
|
13138-33-5
|
98.9%
|
|
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding as...
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T23339 |
SCS
|
3232-36-8
|
98.89%
|
|
SCS is a GABAA receptor antagonist.
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T11277 |
FG 7142
|
78538-74-6
|
98.81%
|
|
FG 7142 (LSU-65) also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 can increase tyrosine hydroxylati...
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T22301 |
L-838417 D9
|
1213669-91-0
|
98.81%
|
|
L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].
|