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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Cat. No. Product name CAS No. Purity Chemical Structure
TN1202 (-)-α-Pinene 7785-26-4 98%

(1S)-(-)-Alpha-Pinene is a natural product

T7794 Zuranolone 1632051-40-1 98%
Zuranolone is an agonist of GABAA receptor.
T11822 LAU159 2055050-87-6 98%
LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
T3318 Wogonoside 51059-44-0 98%
Wogonoside acts as a positive allosteric modulator of the benzodiazepine site of the GABAA receptor.
T15212 Emamectin Benzoate 155569-91-8 98%
Emamectin Benzoate, by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods, acts as ...
T12930 SKF89976A hydrochloride 85375-15-1 98%
SKF89976A hydrochloride is a selective inhibitor of GABA transporter (GAT-1)(IC50s of 0.28 μM, 137.34 μM and 202.8 μM for GAT-1, GAT-2 and GAT-3 in CHO cells, re...
T24381 L-822179 215874-86-5 98%
L-822179 or α5IA is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
TN1217 2'-O-Methylisoliquiritigenin 51828-10-5 98%
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
T28900 T-2000 97846-21-4 98%
T-2000 is a GABA receptor agonist that can be used to study myoclonus and essential tremor.
T23104 Ocinaplon 96604-21-6 98%
GABAA receptors modulator
T22301 L-838417 D9 1213669-91-0 98%
L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].
T11277 FG 7142 78538-74-6 98%
FG 7142 also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 can increase tyrosine hydroxylation and ca...
T23339 SCS 3232-36-8 98%
GABAA receptor antagonist
T38205 3-Aminopropylphosphonic Acid 13138-33-5 98%
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding as...
T11061 DMCM hydrochloride 1215833-62-7 98%
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine. DMCM showed significant differences in human recombinant GABAA αxβ3γ2 receptor sub...
T10618 Broflanilide 1207727-04-5 98%
Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL ...
T7557 Guvacine hydrochloride 6027-91-4 98%
Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
T2775 Baicalin 21967-41-9 98%
Baicalin is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV properties.
T1602 Valproic acid sodium salt 1069-66-5 98%
Valproate Sodium is the sodium salt form of valproic acid with anti-epileptic activity. Valproate sodium is converted into its active form, valproate ion, in blo...
T0883 Tramiprosate 3687-18-1 98%
Because of its similarity in structure to the neurotransmitter gamma-aminobutyric acid (GABA), it has GABAergic effects and may be useful as an anticonvulsant. H...
(-)-α-Pinene
TN1202
<p>(1S)-(-)-Alpha-Pinene is a natural product</p>
Zuranolone
T7794
Zuranolone is an agonist of GABAA receptor.
LAU159
T11822
LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).
Wogonoside
T3318
Wogonoside acts as a positive allosteric modulator of the benzodiazepine site of the GABAA receptor.
Emamectin Benzoate
T15212
Emamectin Benzoate, by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods, acts as ...
SKF89976A hydrochloride
T12930
SKF89976A hydrochloride is a selective inhibitor of GABA transporter (GAT-1)(IC50s of 0.28 μM, 137.34 μM and 202.8 μM for GAT-1, GAT-2 and GAT-3 in CHO cells, re...
L-822179
T24381
L-822179 or α5IA is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
2'-O-Methylisoliquiritigenin
TN1217
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.
T-2000
T28900
T-2000 is a GABA receptor agonist that can be used to study myoclonus and essential tremor.
Ocinaplon
T23104
GABAA receptors modulator
L-838417 D9
T22301
L-838417 is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].
FG 7142
T11277
FG 7142 also modulates GABA-induced chloride flux at GABAA receptors expressing the α1 subunit (EC50= 137 nM). FG 7142 can increase tyrosine hydroxylation and ca...
SCS
T23339
GABAA receptor antagonist
3-Aminopropylphosphonic Acid
T38205
3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding as...
DMCM hydrochloride
T11061
DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine. DMCM showed significant differences in human recombinant GABAA αxβ3γ2 receptor sub...
Broflanilide
T10618
Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL ...
Guvacine hydrochloride
T7557
Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)
Baicalin
T2775
Baicalin is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV properties.
Valproic acid sodium salt
T1602
Valproate Sodium is the sodium salt form of valproic acid with anti-epileptic activity. Valproate sodium is converted into its active form, valproate ion, in blo...
Tramiprosate
T0883
Because of its similarity in structure to the neurotransmitter gamma-aminobutyric acid (GABA), it has GABAergic effects and may be useful as an anticonvulsant. H...
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