T26834 |
BL-1020 Mesylate
|
916898-61-8
|
100%
|
|
BL-1020 Mesylate (CYP-1020 Mesylate) is an orally available GABA A receptor agonist and D2 antagonist that decreases dopamine activity and enhances GABAA activit...
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T27845 |
Losigamone
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112856-44-7
|
100%
|
|
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.
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T20657 |
Muscimol HBr
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18174-72-6
|
100%
|
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Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
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T1673 |
Acamprosate calcium
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77337-73-6
|
|
|
Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.
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T12492 |
Pivagabine
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69542-93-4
|
|
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Pivagabine (CXB-722), a hydrophobic 4-aminobutyric acid derivative, exhibits neuromodulatory activity and successfully penetrates the blood-brain barrier in rats...
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T5880 |
Aminooxyacetic acid hemihydrochloride
|
2921-14-4
|
|
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Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA degrada...
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T16539 |
Piperazine citrate
|
144-29-6
|
|
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Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring. It used as an Anthelmi...
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T2998 |
Dihydromyricetin
|
27200-12-0
|
|
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Dihydromyricetin (Ampelopsin) is a natural antioxidant flavonoid from Ampelopsis grossedentata. Dihydromyricetin is a potent inhibitor of dihydropyrimidinase wit...
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T16489 |
Darigabat
|
1614245-70-3
|
98%
|
|
Darigabat (PF-06372865) is an orally active and selective GABAA receptor modulator that crosses the blood-brain barrier and exhibits anxiolytic activity, with Ki...
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T24381 |
L-822179
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215874-86-5
|
98%
|
|
L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.
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TN1308 |
6-Hydroxyflavanone
|
4250-77-5
|
98%
|
|
6-Hydroxyflavanone, extracted from the leaves of Acorus calamus, exhibits anti-inflammatory and anti-neuropathic pain activity by targeting cyclooxygenase-2 (COX...
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T4993 |
Afloqualone
|
56287-74-2
|
98%
|
|
Afloqualone (HQ-495) is a agonist of GABA Receptor . Target: GABA Receptor in vitro: Afloqualone is a quinazolinone family GABAergic drug. It has sedative and mu...
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T1240 |
Flumazenil
|
78755-81-4
|
98%
|
|
Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous ...
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T37190 |
L-Allylglycine
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16338-48-0
|
98%
|
|
L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo...
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T32098L |
Homocarnosine acetate
|
|
98%
|
|
Homocarnosine acetate is a dipeptide unique to brain consisting of γ-aminobutyric acid (GABA) and histidine. Homocarnosine acetate has antioxidant and anti-infla...
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T8268 |
6,2'-Dihydroxyflavone
|
92439-20-8
|
98%
|
|
6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.
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T28479 |
PZ-II-029
|
164025-44-9
|
98%
|
|
PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.
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T21793 |
CGP 35348
|
123690-79-9
|
98%
|
|
CGP 35348 is a selective antagonist of GABAB receptor (EC50 = 34 μM). CGP 35348 can be used in studies of neuromuscular coordination and spatial learning after n...
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