T13803 |
N-Oleoyl glycine
|
2601-90-3
|
99.92%
|
|
N-Oleoyl Glycine, a Lipoamino Acid, Stimulates Adipogenesis Associated With Activation of CB1 Receptor and Akt Signaling Pathway in 3T3-L1 Adipocyte
|
T21450 |
AM-2232
|
335161-19-8
|
99.89%
|
|
AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.
|
T6527 |
GW842166X
|
666260-75-9
|
99.88%
|
|
GW842166X is a potent and highly selective agonist of cannabinoid receptor CB2 receptor with EC50 of 63 nM, shows no significant activity at CB1 receptor. Phase ...
|
TP1939L1 |
RVD-Hpα acetate(1193362-76-3 free base)
|
TP1939L1
|
99.87%
|
|
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. Increases intracellular Ca2+ levels in cell...
|
T39024 |
PrNMI
|
1541244-33-0
|
99.87%
|
|
PrNMI is a highly effective and orally active agonist targeting the peripherally restricted cannabinoid 1 receptor (CB1R). It exhibits pronounced analgesic prope...
|
TP1900L1 |
Hemopressin (human, mouse) acetate
|
TP1900L1
|
99.86%
|
|
Hemopressin (human, mouse) acetate is a nonapeptide derived from the α1-chain of hemoglobin, is originally isolated from rat brain homogenates. Hemopressin is or...
|
T14204 |
6-Iodopravadoline
|
164178-33-0
|
99.86%
|
|
6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.
|
T41350 |
6-Bromopravadoline
|
166599-63-9
|
99.84%
|
|
6-Bromopravadoline (WIN 54461) (WIN 54461) is an antagonist of CB1. 6-Bromopravadoline acts as an inhibitor of the binding of [3H]Win 55212-2 (IC 50 =515 nM) ref...
|
T4654 |
(±)-Ibipinabant
|
362519-49-1
|
99.83%
|
|
(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.
|
TN2268 |
Tetrahydromagnolol
|
20601-85-8
|
99.82%
|
|
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
|
T7705 |
GW 405833
|
180002-83-9
|
99.82%
|
|
GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective
|
T21861 |
Drinabant
|
358970-97-5
|
99.8%
|
|
Drinabant (AVE-1625) is an orally active CB1 receptor antagonist. Drinabant inhibits the agonist-stimulated calcium signal with IC50 values of 25 nM and 10 nM fo...
|
T22103 |
ML-193
|
713121-80-3
|
99.79%
|
|
ML-193 (CID 1261822) is a potent and selective GPR55 antagonist( IC50 : 221 nM). It shows more than 27-fold selectivity for GPR55 over GPR35, CB1 and CB2, and ca...
|
T33452 |
ML192
|
460331-61-7
|
99.79%
|
|
ML192 (CID1434953) is a selective GPR55 ligand antagonist. ML192 is an inhibitor that inhibits β-arrestin transport, ERK1/2 phosphorylation, and PKCβII transloca...
|
TC0019 |
Pregnenolone acetate
|
1778-02-5
|
99.78%
|
|
Pregnenolone acetate is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones. It acts as a signaling-specific inhibi...
|
T3736 |
Olivetol
|
500-66-3
|
99.74%
|
|
Olivetol (5-n-Amylresorcinol) (5-pentylresorcinol, 5-pentyl-1,3-benzenediol) is an organic compound found in certain species of lichen; it is also a precursor in...
|
T22114 |
NESS 0327
|
494844-07-4
|
99.74%
|
|
NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.
|
T12306 |
OMDM-5
|
616884-66-3
|
99.72%
|
|
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
|
T16928 |
SR144528
|
192703-06-3
|
99.6%
|
|
SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).
|
T4478 |
CID 16020046
|
834903-43-4
|
99.59%
|
|
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
|