Home Tools
Log in
Cart

Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TMA1012 Ganoderiol F 114567-47-4 98%
Ganoderiol F
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
T19449 N-desmethyl Enzalutamide D6 T19449 98%
N-desmethyl Enzalutamide D6
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
T0380 Bicalutamide 90357-06-5 99.97%
Bicalutamide
Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the ...
T2339 Apalutamide 956104-40-8 99.97%
Apalutamide
Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T68020 Zanoterone 107000-34-0 99.96%
Zanoterone
Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary disorders and oncological disorders and m...
T0419 Testosterone propionate 57-85-2 99.92%
Testosterone propionate
Testosterone Propionate is a short acting oil-based injectable formulation of testosterone. Testosterone inhibits gonadotropin secretion from the pituitary gland...
T0489 Flutamide 13311-84-7 99.92%
Flutamide
Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent and canine species.
T1541 Drospirenone 67392-87-4 99.85%
Drospirenone
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T9179 CLP-3094 312749-73-8 99.84%
CLP-3094
CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activi...
TN1370 Allura Red AC 25956-17-6 99.82%
Allura Red AC
Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes suscept...
T0856 Dehydroisoandrosterone 3-acetate 853-23-6 99.81%
Dehydroisoandrosterone 3-acetate
Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.
TQ0209 Ailanthone 981-15-7 99.78%
Ailanthone
Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR sp...
T2236 RU 58841 154992-24-2 99.77%
RU 58841
RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.
T16090 MK-0773 606101-58-0 99.63%
MK-0773
MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.
T13272 UT-155 2031161-35-8 99.63%
UT-155
UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).
T0476 Spironolactone 52-01-7 99.63%
Spironolactone
Spironolactone (SC9420) is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
T6509 Galeterone 851983-85-2 99.57%
Galeterone
Galeterone (VN 124) is an orally bioavailable small-molecule androgen receptor modulator and CYP17 lyase inhibitor with potential antiandrogen activity. Galetero...
T2321 Protodioscin 55056-80-9 99.56%
Protodioscin
Protodioscin (Furostanol I) is a major steroidal saponin in dioscoreae rhizome, with anti-hyperlipidemia, anti-cancer properties.
T12928 SK33 1928724-23-5 99.55%
SK33
SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity.
T14116 ACP-105 899821-23-9 99.53%
ACP-105
ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testostero...
Ganoderiol F
TMA1012
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
N-desmethyl Enzalutamide D6
T19449
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
Bicalutamide
T0380
Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the ...
Apalutamide
T2339
Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
Zanoterone
T68020
Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary disorders and oncological disorders and m...
Testosterone propionate
T0419
Testosterone Propionate is a short acting oil-based injectable formulation of testosterone. Testosterone inhibits gonadotropin secretion from the pituitary gland...
Flutamide
T0489
Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent and canine species.
Drospirenone
T1541
Drospirenone (ZK 3059) is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
CLP-3094
T9179
CLP-3094 (2-([2-(4-CHLOROPHENOXY)ETHYL]THIO)-1H-BE) is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activi...
Allura Red AC
TN1370
Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes suscept...
Dehydroisoandrosterone 3-acetate
T0856
Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.
Ailanthone
TQ0209
Ailanthone (Δ13-Dehydrochaparrinone) is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR sp...
RU 58841
T2236
RU 58841 (PSK-3841) is a specific androgen receptor antagonist or anti-androgen; RU 58841(PSK-3841) has a significant effect on hair regrowth.
MK-0773
T16090
MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.
UT-155
T13272
UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).
Spironolactone
T0476
Spironolactone (SC9420) is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
Galeterone
T6509
Galeterone (VN 124) is an orally bioavailable small-molecule androgen receptor modulator and CYP17 lyase inhibitor with potential antiandrogen activity. Galetero...
Protodioscin
T2321
Protodioscin (Furostanol I) is a major steroidal saponin in dioscoreae rhizome, with anti-hyperlipidemia, anti-cancer properties.
SK33
T12928
SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity.
ACP-105
T14116
ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testostero...
1 2 3 4 5 6
TargetMol