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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T8348 Phentolamine 50-60-2 99.86%
Phentolamine
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T0993 Methoxamine hydrochloride 61-16-5 99.86%
Methoxamine hydrochloride
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T6466 Dexmedetomidine hydrochloride 145108-58-3 99.86%
Dexmedetomidine hydrochloride
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE,...
T0505 Methyldopa 555-30-6 99.86%
Methyldopa
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic...
T1496 Amiodarone hydrochloride 19774-82-4 99.85%
Amiodarone hydrochloride
Amiodarone hydrochloride (Amiodarone HCl) is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action ...
T8738 LUN42518 HCl 47142-51-8(free base) 99.85%
LUN42518 HCl  47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
T0469 Octopamine hydrochloride 770-05-8 99.85%
Octopamine hydrochloride
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a ne...
T3275 Nefazodone hydrochloride 82752-99-6 99.85%
Nefazodone hydrochloride
Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.
T40622 Mapenterol hydrochloride 54238-51-6 99.85%
Mapenterol hydrochloride
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
T22316 Doxazosin 74191-85-8 99.85%
Doxazosin
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
T0154 Nebivolol hydrochloride 152520-56-4 99.85%
Nebivolol hydrochloride
Nebivolol hydrochloride (R 065824 hydrochloride) is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR throug...
T30140 Arotinolol hydrochloride 68377-91-3 99.84%
Arotinolol hydrochloride
Arotinolol hydrochloride(Arotinolol HCl) is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I...
T7044 Norepinephrine 51-41-2 99.84%
Norepinephrine
Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression ...
T0115 Idazoxan hydrochloride 79944-56-2 99.84%
Idazoxan hydrochloride
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0042 Xylometazoline hydrochloride 1218-35-5 99.83%
Xylometazoline hydrochloride
Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.
T6422 Brimonidine Tartrate 70359-46-5 99.83%
Brimonidine Tartrate
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pres...
T0277 Metaproterenol hemisulfate 5874-97-5 99.83%
Metaproterenol hemisulfate
Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
T23382 Spiroxatrine 1054-88-2 99.83%
Spiroxatrine
Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2,...
T23557 Talibegron hydrochloride 178600-17-4 99.82%
Talibegron hydrochloride
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Re...
T5S2178 Fargesin 31008-19-2 99.82%
Fargesin
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Far...
Phentolamine
T8348
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
Methoxamine hydrochloride
T0993
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
Dexmedetomidine hydrochloride
T6466
Dexmedetomidine hydrochloride (Precedex) is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE,...
Methyldopa
T0505
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic...
Amiodarone hydrochloride
T1496
Amiodarone hydrochloride (Amiodarone HCl) is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action ...
LUN42518 HCl 47142-51-8(free base)
T8738
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
Octopamine hydrochloride
T0469
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a ne...
Nefazodone hydrochloride
T3275
Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.
Mapenterol hydrochloride
T40622
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
Doxazosin
T22316
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
Nebivolol hydrochloride
T0154
Nebivolol hydrochloride (R 065824 hydrochloride) is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR throug...
Arotinolol hydrochloride
T30140
Arotinolol hydrochloride(Arotinolol HCl) is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I...
Norepinephrine
T7044
Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression ...
Idazoxan hydrochloride
T0115
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
Xylometazoline hydrochloride
T0042
Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.
Brimonidine Tartrate
T6422
Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pres...
Metaproterenol hemisulfate
T0277
Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
Spiroxatrine
T23382
Spiroxatrine (R 5188) is a selective and potent 5-HT1α and α2-adrenergic dual antagonist with sedative activity and inhibitory effects on 5-HT1α, 5-HT1 β, 5-HT2,...
Talibegron hydrochloride
T23557
Talibegron hydrochloride (ZD2079 hydrochloride) is an β3 adrenergic receptor agonist with a pD2 of 3.72 on phenylephrine-preconstricted rat mesenteric artery. Re...
Fargesin
T5S2178
1. Fargesin ((+/-)-Fargesin) as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Far...
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TargetMol