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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T21787L Azepexole hydrochloride 147663-20-5 98.03%
Azepexole hydrochloride
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
T1045 Trimipramine maleate 521-78-8 98.02%
Trimipramine maleate
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
T6860 (RS)-ICI-118551 Hydrochloride 1217094-53-5 98.02%
(RS)-ICI-118551 Hydrochloride
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
T21371 Apraclonidine hydrochloride 73218-79-8 98.01%
Apraclonidine hydrochloride
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pre...
T1287 Synephrine 94-07-5 98%
Synephrine
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T1504 Silodosin 160970-54-7 98%
Silodosin
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
T1459 Cisatracurium besylate 96946-42-8 98%
Cisatracurium besylate
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T0365 Thioridazine hydrochloride 130-61-0 98%
Thioridazine hydrochloride
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selecti...
T3158 Harmane 486-84-0 97.89%
Harmane
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T11726 JP1302 dihydrochloride 1259314-65-2 97.83%
JP1302 dihydrochloride
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a...
T12596 (4E)-SUN9221 222318-55-0 97.79%
(4E)-SUN9221
(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in hypertens...
T3046 BMY 7378 dihydrochloride 21102-95-4 97.67%
BMY 7378 dihydrochloride
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T0446 Naphazoline hydrochloride 550-99-2 97.6%
Naphazoline hydrochloride
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
T68164 Tolamolol 38103-61-6 97.58%
Tolamolol
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the trea...
T70047 Bedoradrine 194785-19-8 97.53%
Bedoradrine
Bedoradrine free base is a novel, highly selective β2-adrenoceptor agonist for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
T21447 Tolazoline 59-98-3 97.51%
Tolazoline
Tolazoline (Benzalolin), a non-selective competitive α-adrenergic receptor antagonist, is used as a vasodilator to treat spasms of peripheral blood vessels. It h...
T28829 Soquinolol 61563-18-6 97.48%
Soquinolol
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long durat...
T68114L Nardeterol HCl 97.36%
Nardeterol HCl
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4
T10812 Cicloprolol hydrochloride 63686-79-3 97.26%
Cicloprolol hydrochloride
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
T77641 5-Bromoimidazo[1,2-A]Pyrazine 87597-26-0 97.04%
5-Bromoimidazo[1,2-A]Pyrazine
5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.
Azepexole hydrochloride
T21787L
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
Trimipramine maleate
T1045
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
(RS)-ICI-118551 Hydrochloride
T6860
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
Apraclonidine hydrochloride
T21371
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist. Apraclonidine hydrochloride lowers intraocular pre...
Synephrine
T1287
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
Silodosin
T1504
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
Cisatracurium besylate
T1459
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Thioridazine hydrochloride
T0365
Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selecti...
Harmane
T3158
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
JP1302 dihydrochloride
T11726
JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Ki (binding affinity) value of 28 nM and a...
(4E)-SUN9221
T12596
(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in hypertens...
BMY 7378 dihydrochloride
T3046
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
Naphazoline hydrochloride
T0446
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Tolamolol
T68164
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the trea...
Bedoradrine
T70047
Bedoradrine free base is a novel, highly selective β2-adrenoceptor agonist for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
Tolazoline
T21447
Tolazoline (Benzalolin), a non-selective competitive α-adrenergic receptor antagonist, is used as a vasodilator to treat spasms of peripheral blood vessels. It h...
Soquinolol
T28829
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a long durat...
Nardeterol HCl
T68114L
Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4
Cicloprolol hydrochloride
T10812
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
5-Bromoimidazo[1,2-A]Pyrazine
T77641
5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.
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TargetMol