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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T6519 Gramine 87-52-5 98.44%
Gramine
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
T68124 Pafenolol 75949-61-0 98.43%
Pafenolol
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.
T26778L Besipirdine hydrochloride 130953-69-4 98.40%
Besipirdine hydrochloride
Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine hydrochloride inhib...
T7079 Batefenterol 743461-65-6 98.4%
Batefenterol
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
T17111 Todralazine hydrochloride 3778-76-5 98.32%
Todralazine hydrochloride
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can b...
T11095L DREADD agonist 21 56296-18-5 98.27%
DREADD agonist 21
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
T6653 Salmeterol Xinafoate 94749-08-3 98.24%
Salmeterol Xinafoate
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma sympto...
T28895 T-0509 96843-99-1 98.21%
T-0509
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-adrenoceptor...
T33386 Milveterol HCl 804518-03-4 98.2%
Milveterol HCl
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
T10250 ADRA1D receptor antagonist 1 HCl 1191908-14-1 98.13%
ADRA1D receptor antagonist 1 HCl
ADRA1D receptor antagonist 1 HCl is an orally active, potent and selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activ...
T68023L Tolnapersine TFA T68023L 98.10%
Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
T11148 Ecastolol 77695-52-4 98.1%
Ecastolol
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
TN7129 Methyl maslinate 22425-82-7 98.1%
Methyl maslinate
Methyl maslinate (Maslinic acid methyl ester) is an antagonist of β- adrenergic receptor with cardiotonic and antidysrhythmic properties. Methyl maslinate can be...
T0397 Tetrahydrozoline 84-22-0 98.07%
Tetrahydrozoline
Tetrahydrozoline (Tetryzoline), an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of th...
T23301 (S)-(+)-Niguldipine hydrochloride 113145-69-0 98.06%
(S)-(+)-Niguldipine hydrochloride
(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
TP1902L1 G-Protein antagonist peptide acetate TP1902L1 98.06%
G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide aceta...
T1158 Phenoxybenzamine hydrochloride 63-92-3 98.04%
Phenoxybenzamine hydrochloride
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...
T21787L Azepexole hydrochloride 147663-20-5 98.03%
Azepexole hydrochloride
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
T1045 Trimipramine maleate 521-78-8 98.02%
Trimipramine maleate
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
T6860 (RS)-ICI-118551 Hydrochloride 1217094-53-5 98.02%
(RS)-ICI-118551 Hydrochloride
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
Gramine
T6519
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4...
Pafenolol
T68124
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.
Besipirdine hydrochloride
T26778L
Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine hydrochloride inhib...
Batefenterol
T7079
Batefenterol (TD-5959) (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic an...
Todralazine hydrochloride
T17111
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can b...
DREADD agonist 21
T11095L
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
Salmeterol Xinafoate
T6653
Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma sympto...
T-0509
T28895
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-adrenoceptor...
Milveterol HCl
T33386
Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
ADRA1D receptor antagonist 1 HCl
T10250
ADRA1D receptor antagonist 1 HCl is an orally active, potent and selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) with potential antiproliferative activ...
Tolnapersine TFA
T68023L
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Ecastolol
T11148
Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
Methyl maslinate
TN7129
Methyl maslinate (Maslinic acid methyl ester) is an antagonist of β- adrenergic receptor with cardiotonic and antidysrhythmic properties. Methyl maslinate can be...
Tetrahydrozoline
T0397
Tetrahydrozoline (Tetryzoline), an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of th...
(S)-(+)-Niguldipine hydrochloride
T23301
(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
G-Protein antagonist peptide acetate
TP1902L1
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide aceta...
Phenoxybenzamine hydrochloride
T1158
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihyp...
Azepexole hydrochloride
T21787L
Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic ...
Trimipramine maleate
T1045
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepineph...
(RS)-ICI-118551 Hydrochloride
T6860
ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors...
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TargetMol