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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T3232 Higenamine hydrochloride 11041-94-4 98.75%
Higenamine hydrochloride
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class...
T3431 Pardoprunox hydrochloride 269718-83-4 98.73%
Pardoprunox hydrochloride
Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) an...
T11015 Midaglizole hydrochloride 79689-25-1 98.73%
Midaglizole hydrochloride
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenocepto...
T77566 (3aR,9aR)-Fluparoxan 105182-47-6 98.68%
(3aR,9aR)-Fluparoxan
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
T60773 Butofilolol 58930-32-8 98.68%
Butofilolol
Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.
T10066 2',5'-Dideoxyadenosine 6698-26-6 98.66%
2',5'-Dideoxyadenosine
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
T24579 Oxyfedrine L-form HCl 16777-42-7 98.66%
Oxyfedrine L-form HCl
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.
T0248 Clorprenaline hydrochloride 6933-90-0 98.65%
Clorprenaline hydrochloride
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
T14490 Talipexole dihydrochloride 36085-73-1 98.64%
Talipexole dihydrochloride
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
T22612 BMY-14802 hydrochloride 105565-55-7 98.64%
BMY-14802 hydrochloride
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
T20157 Brimonidine 59803-98-4 98.60%
Brimonidine
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
T5471 GUANABENZ 5051-62-7 98.6%
GUANABENZ
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T26778 Besipirdine 119257-34-0 98.59%
Besipirdine
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine inhibits volta...
T22369 Midodrine 42794-76-3 98.57%
Midodrine
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
T13804 OPC-28326 167626-17-7 98.56%
OPC-28326
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
T31175 Dabelotine 118976-38-8 98.55%
Dabelotine
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
T8149 Dobutamine hydrochloride 49745-95-1 98.52%
Dobutamine hydrochloride
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T26923 Bunazosin Hydrochloride 52712-76-2 98.48%
Bunazosin Hydrochloride
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
T10952 Dabuzalgron 219311-44-1 98.47%
Dabuzalgron
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
T6562 Latrepirdine dihydrochloride 97657-92-6 98.45%
Latrepirdine dihydrochloride
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
Higenamine hydrochloride
T3232
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class...
Pardoprunox hydrochloride
T3431
Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1) an...
Midaglizole hydrochloride
T11015
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenocepto...
(3aR,9aR)-Fluparoxan
T77566
(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental diso...
Butofilolol
T60773
Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.
2',5'-Dideoxyadenosine
T10066
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
Oxyfedrine L-form HCl
T24579
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.
Clorprenaline hydrochloride
T0248
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
Talipexole dihydrochloride
T14490
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and intestinal...
BMY-14802 hydrochloride
T22612
BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects. BMY-14802 hydrochloride is...
Brimonidine
T20157
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P. It is used to treat open-angle glaucoma or ocular hypertensi...
GUANABENZ
T5471
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
Besipirdine
T26778
Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic and cardiovascular activities.Besipirdine inhibits volta...
Midodrine
T22369
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
OPC-28326
T13804
OPC-28326 is a specific an α2-adrenergic receptor antagonist and acts as a peripheral vasodilator. OPC-28326 inhibits α2A-, α2B- and α2C-adrenoceptors with Ki of...
Dabelotine
T31175
Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.
Dobutamine hydrochloride
T8149
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
Bunazosin Hydrochloride
T26923
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
Dabuzalgron
T10952
Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxicit...
Latrepirdine dihydrochloride
T6562
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
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TargetMol