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Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma, for example.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TCS2185 Yohimbine 146-48-5
Yohimbine
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T1769 Pardoprunox 269718-84-5
Pardoprunox
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials st...
TN4882 Quinine HCl 130-89-2 98%
Quinine HCl
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T5450 DL-071-IT 55104-39-7 98%
DL-071-IT
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist. DL-071-IT showed intrinsic sympathomimetic activity and weak membrane ...
T13470 (±)-Levomepromazine-d6 1189805-51-3 98%
(±)-Levomepromazine-d6
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T78567 Moprolol 5741-22-0 98%
Moprolol
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].
T79641 (±)-N-Methylcoclaurine 1472-62-4 98%
(±)-N-Methylcoclaurine
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
T80175 Conopeptide rho-TIA 381725-58-2 98%
Conopeptide rho-TIA
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive i...
T80477 Muscarinic toxin 3 873336-87-9 98%
Muscarinic toxin 3
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 f...
TN1797 Isorhoifolin 552-57-8 98%
Isorhoifolin
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
T81798 Mibenratide TFA 98%
Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].
T15042 D2343 72734-63-5 98%
D2343
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T6663 Scopine hydrochloride 85700-55-6 98%
Scopine hydrochloride
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acu...
T16769 Ro 363 74513-77-2 98%
Ro 363
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
TN2267 Tetrahydroalstonine 6474-90-4 98%
Tetrahydroalstonine
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
TN3368 Akuammigine 642-17-1 98%
Akuammigine
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T11786 KUL-7211 racemate 911196-40-2 98%
KUL-7211 racemate
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
T12815 (S)-Terazosin 109351-33-9 98%
(S)-Terazosin
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
T13285 Vatinoxan hydrochloride 130466-38-5 98%
Vatinoxan hydrochloride
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
T6562 Latrepirdine dihydrochloride 97657-92-6 98%
Latrepirdine dihydrochloride
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
Yohimbine
TCS2185
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
Pardoprunox
T1769
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials st...
Quinine HCl
TN4882
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
DL-071-IT
T5450
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist. DL-071-IT showed intrinsic sympathomimetic activity and weak membrane ...
(±)-Levomepromazine-d6
T13470
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
Moprolol
T78567
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].
(±)-N-Methylcoclaurine
T79641
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
Conopeptide rho-TIA
T80175
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive i...
Muscarinic toxin 3
T80477
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 f...
Isorhoifolin
TN1797
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
Mibenratide TFA
T81798
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].
D2343
T15042
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
Scopine hydrochloride
T6663
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acu...
Ro 363
T16769
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
Tetrahydroalstonine
TN2267
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
KUL-7211 racemate
T11786
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
(S)-Terazosin
T12815
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
Vatinoxan hydrochloride
T13285
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
Latrepirdine dihydrochloride
T6562
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets, including histamine receptors,...
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TargetMol