TCS2185 |
Yohimbine
|
146-48-5
|
|
|
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
|
T1769 |
Pardoprunox
|
269718-84-5
|
|
|
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials st...
|
TN4882 |
Quinine HCl
|
130-89-2
|
98%
|
|
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
|
T5450 |
DL-071-IT
|
55104-39-7
|
98%
|
|
DL-071-IT (Afurolol Hydrochloride) is a potent non-selective beta-adrenoceptor antagonist. DL-071-IT showed intrinsic sympathomimetic activity and weak membrane ...
|
T13470 |
(±)-Levomepromazine-d6
|
1189805-51-3
|
98%
|
|
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
|
T78567 |
Moprolol
|
5741-22-0
|
98%
|
|
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].
|
T79641 |
(±)-N-Methylcoclaurine
|
1472-62-4
|
98%
|
|
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
|
T80175 |
Conopeptide rho-TIA
|
381725-58-2
|
98%
|
|
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive i...
|
T80477 |
Muscarinic toxin 3
|
873336-87-9
|
98%
|
|
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57 f...
|
TN1797 |
Isorhoifolin
|
552-57-8
|
98%
|
|
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile f...
|
T81798 |
Mibenratide TFA
|
|
98%
|
|
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].
|
T15042 |
D2343
|
72734-63-5
|
98%
|
|
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
|
T6663 |
Scopine hydrochloride
|
85700-55-6
|
98%
|
|
Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acu...
|
T16769 |
Ro 363
|
74513-77-2
|
98%
|
|
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial contr...
|
TN2267 |
Tetrahydroalstonine
|
6474-90-4
|
98%
|
|
Tetrahydroalstonine is an indole alkaloid extracted from the fruit of Rhazya stricta and is a selective α2-adrenoceptor antagonist. tetrahydroalstonine has shown...
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
T11786 |
KUL-7211 racemate
|
911196-40-2
|
98%
|
|
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211.
|
T12815 |
(S)-Terazosin
|
109351-33-9
|
98%
|
|
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with...
|
T13285 |
Vatinoxan hydrochloride
|
130466-38-5
|
98%
|
|
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
|
T11036 |
Diacetolol D7
|
1346604-19-0
|
98%
|
|
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
|