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sb216469

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
Upidosin
SB-216469, SB 216469, Rec 15-2739, Recordati 15 2739
T9762152735-23-4
Upidosin (SB-216469) is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM.
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