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Search Result

Search Results for " non-nmda "

Targets

iGluR

19

Compounds

3

Natural Products

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T8458 CNQX disodium iGluR
CNQX disodium is a competitive non-NMDA receptor antagonist and competitive AMPA/kainate receptor antagonist in neuronal cultures.
T8459 DNQX disodium salt DNQX Disodium NMDAR , iGluR
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor
T7304 DNQX FG 9041 GluR , iGluR
DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)
T7178 CNQX FG9065 GluR , iGluR
CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)
T2362 QNZ46 NMDAR , iGluR
QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.
T26645 Aptiganel CNS 1102,CNS-1102,CNS1102 NMDAR
Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.
T23048 N20C hydrochloride 2-((3,3-diphenylpropyl)amino)acetamide hydrochloride NMDAR
N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.
T22798 Gavestinel GV 150526,Gavestinel sodium salt NMDAR , iGluR
Gavestinel (GV 150526) is a non-competitive NMDA receptor antagonist that is potent, selective and orally active.Gavestinel binds to the glycine site of the NMDA receptor with a binding affinity (pKi value) of 8.5.Gavest...
T6352 (-)-Dizocilpine maleate C13737,(-)-MK 801 (Maleate),(-)-MK 801 Maleate NMDAR , iGluR
(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.
T1751 Eliprodil SL-820715 NMDAR , iGluR
Eliprodil (SL-820715)(SL-820715), a non-competitive NR2B-NMDA receptor antagonist(IC50: 1 uM), less effective for NR2A- and NR2C-containing receptors(IC50> 100 uM). It has been used in trials studying the treatment of Pa...
T22513 4-PPBP maleate Sigma receptor , NMDAR
4-PPBP maleate is a potent σ1 receptor (ligand) agonist. 4-PPBP maleate can be considered a selective, non-competitive NR1a/2B NMDA receptor antagonist in the context of Xenopus oocytes expression. 4-PPBP maleate has neu...
T6504 Flupirtine maleate Katadolon maleate Potassium Channel , NMDAR , iGluR
Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. It is an NMDA receptor antagonist , and also a specific neuronal potassium channel opener.
T22640 CCMQ Others
inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites
T61470 NMDA receptor antagonist 5
NMDA receptor antagonist 5 (Compound 10e), a potent and non-toxic NMDA receptor antagonist, exhibits brain permeability. It is of significance in studying neurological disorders [1].
TP2235 Conantokin-T Others
Non-competitive NMDA receptor antagonist
T21449 GYKI-52466 GYKI 52,466,GYKI-5,2466,GYKI52,466
GYKI-52466 is a selective non-competitive AMPA receptor antagonist (IC50 values are 10-20, ~ 450 and >50 μM for AMPA-, kainate- and NMDA-induced responses, respectively) used as a Skeletal muscle relaxant, orally active ...
T11522 GYKI 52466 dihydrochloride Others
GYKI 52466 dihydrochloride is orally active and non-competitive kainate- and AMPA-activated currents antagonist (IC50s: 7.5 μM and 11 μM). It is inactive against NMDA or γ-aminobutyric acid responses. It is a muscle rela...
T69422 Flupirtine HCl
Flupirtine HCl is the salt form of Flupirtine, also known as W-2964, an aminopyridine that functions as a centrally acting non-opioid analgesic. It first became available in Europe in 1984, and is sold mainly under the n...
T37671 CAY10608 CAY10608
N-Methyl-D-aspartate (NMDA) receptors are Ca2+ permeable ligand-gated channels of the central nervous system that are activated after binding of the co-agonists glutamate and glycine. CAY10608 is a propanolamine that pot...
Cat No. Product Name Synonyms Targets
T3377 L-Phenylalanine (S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine Calcium Channel , Endogenous Metabolite , iGluR
L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.
T6S0659 Rhynchophylline Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin Calcium Channel , NF-κB
1. Rhynchophylline (Mitrinermine) can protect against ischemic damage, probably via regulating the Akt/mTOR pathway. 2. Rhynchophylline can protect against glutamate-induced neuronal death, can inhibit MA impairment in c...
T2O2728 Glycine 2-Aminoacetic acid,Glycolixir,Aminoacetic acid,Glycosthene,Glycocoll MT Receptor , Endogenous Metabolite , iGluR
glycine (2-Aminoacetic acid) is a non-essential amino acid. It is found primarily in gelatin and silk fibroin and used therapeutically as a nutrient. It is also a fast inhibitory neurotransmitter.

Natural Products

L-Phenylalanine
T3377
Synonym: (S)-2-Amino-3-phenylpropionic acid,phenylalanine,3-Phenyl-L-alanine
Target: Calcium Channel, Endogenous Metabolite, iGluR
Rhynchophylline
T6S0659
Synonym: Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
glycine
T2O2728
Synonym: 2-Aminoacetic acid,Glycolixir,Aminoacetic acid,Glycosthene,Glycocoll
Target: MT Receptor, Endogenous Metabolite, iGluR

Recombinant Proteins

Species：
Human (1)
Mouse (1)
Expression System：
Baculovirus-Insect Cells (2)
Tag：
His,GST (2)
Cat No. Product Name Species Expression System
TMPY-04384 Src Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
Proto-oncogene tyrosine-protein kinase SRC is a hydrophobic protein belonging to the SRC family kinase including nine members that is a family of non-receptor tyrosine kinases. SRC protein may exist in different forms: C...
TMPY-04434 Src Protein, Mouse, Recombinant (His & GST) Mouse Baculovirus-Insect Cells
Proto-oncogene tyrosine-protein kinase SRC is a hydrophobic protein belonging to the SRC family kinase including nine members that is a family of non-receptor tyrosine kinases. SRC protein may exist in different forms: C...
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