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Results for "
difelikefalin hydrochloride
" in TargetMol Product Catalog- Inhibitors & Agonists2
- Isotope Products1
Difelikefalin HCl
T695372711717-77-8
Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin HCl is selective for KOR over the μ-opioid receptor (MOR; EC50 = >1 µM in a transactivation assay). It reduces acetic acid-induced writhing, as well as scratching behavior induced by the KOR antagonist GNTI, in mice (ED50s = 0.07 and 0.05 mg/kg, respectively).
- $1,970
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Difelikefalin-d5
T212328
Difelikefalin-d5 (CR-845-d5) hydrochloride is the deuterated form of Difelikefalin. Difelikefalin (CR-845) acts as a selective κ-opioid receptor (KOR) agonist. It exhibits anti-inflammatory properties and shows potential for managing itch associated with conditions such as chronic kidney disease.
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