TP1572 |
GR-73632
|
133156-06-6
|
99.68%
|
|
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
|
T3034 |
Eprazinone dihydrochloride
|
10402-53-6
|
99.25%
|
|
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
|
T7631L |
Eledoisin Related Peptide 2TFA
|
T7631L
|
99%
|
|
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.
|
T13329L |
Vofopitant dihydrochloride
|
168266-51-1
|
98.99%
|
|
Vofopitant dihydrochloride (GR 205171A) is an orally available, selective tachykinin NK1 receptor antagonist that inhibits [3H]SP binding to NK1 with pKi values ...
|
T15278 |
Fezolinetant
|
1629229-37-3
|
98.62%
|
|
Fezolinetant (ESN-364) is an antagonist of the neurokinin 3 receptor (NK3R). It is used for the treatment of menopausal hot flushes.
|
TP2227L |
C14TKL-1 acetate
|
TP2227L
|
98.56%
|
|
C14TKL-1 acetate is a NK1 receptor agonist.
|
TP1363L |
Neurokinin B acetate(86933-75-7 free base)
|
TP1363L
|
98.53%
|
|
Neurokinin B acetate(86933-75-7 free base) is the acetate form of Neurokinin B, which belongs to the tachykinin family. Neurokinin binds to neurokinin receptor 1...
|
T3724 |
Rolapitant hydrochloride
|
858102-79-1
|
98.46%
|
|
Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a K i of 0.66 nM. Rolapita...
|
TP1772L |
Hemokinin 1 (mouse) acetate(208041-90-1 free base)
|
TP1772L
|
98.33%
|
|
Hemokinin 1 (mouse) acetate is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 recep...
|
TP1087 |
Substance P
|
33507-63-0
|
98%
|
|
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.
|
T7549 |
Talnetant
|
174636-32-9
|
98%
|
|
Talnetant (SB 223412) is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic ...
|
T7209 |
Maropitant
|
147116-67-4
|
98%
|
|
Maropitant is a selective neurokinin (NK1) receptor antagonist.
|
T22811L |
GR 94800 acetate
|
|
97.86%
|
|
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
|
TP1899L1 |
Hemokinin 1 (human) acetate(491851-53-7 free base)
|
TP1899L1
|
97.82%
|
|
Hemokinin 1 (human) acetate is an endogenous substance P homolog that is a selective agonist at the tachykinin NK1 receptor (IC50 values are 1.8, 370 and 480 nM ...
|
T13329 |
Vofopitant
|
168266-90-8
|
97.61%
|
|
Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).
|
T1790 |
Fosaprepitant dimeglumine
|
265121-04-8
|
97.39%
|
|
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic act...
|
T68068L |
(R)-CJ 11974
|
187281-35-2
|
97.03%
|
|
(R)-CJ 11974 is a novel non-peptide neurokinin NK1 substance P receptor antagonist with potential analgesic activity that can be used to study chemotherapy-induc...
|
T68068 |
Ezlopitant
|
147116-64-1
|
97.03%
|
|
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.
|
TP1862L |
[Sar9] Substance P acetate(77128-75-7 free base)
|
TP1862L
|
96.67%
|
|
[Sar9]-Substance P acetate is one of NK-1 receptor agonist. The action of SP on progesterone metabolism was mimicked by the rNK1-specific agonist [Sar-9,Met(O2)1...
|
TP1738L |
Kassinin acetate(63968-82-1 free base)
|
TP1738L
|
95.81%
|
|
Kassinin acetate is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides.
|