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Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T30098 Aplindore Fumarate 189681-71-8 100%
Aplindore Fumarate
Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors,...
T1735 Lurasidone hydrochloride 367514-88-3 100%
Lurasidone hydrochloride
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotoni...
T4262 BisfluoroModafinil 90280-13-0
BisfluoroModafinil
CRL-40940 is a selective dopaminergic reuptake inhibitor
T8653 DOPEXAMINE 86197-47-9
DOPEXAMINE
Dopexamine is a dopaminergic agonist
T14767 BP 897 hydrochloride 314776-92-6
BP 897 hydrochloride
BP 897 is a potent and selective agonist of dopamine D3 receptor and it is a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 re...
T15270 Fananserin 127625-29-0 98%
Fananserin
Fananserin is an effective, selective and oral active antagonist of 5-HT2 (Ki = 0.37 nM for the rat 5-HT2A). Fananserin is an antagonist of human D4 receptor (Ki...
T1211 Levosulpiride 23672-07-3 98%
Levosulpiride
Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
T0338 Minaprine 25905-77-5 98%
Minaprine
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
T8385 Metoclopramide hydrochloride hydrate 54143-57-6 98%
Metoclopramide hydrochloride hydrate
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It...
T13164 Tipepidine hydrochloride 1449686-84-3 98%
Tipepidine hydrochloride
Tipepidine hydrochloride is a reversible inhibitor of dopamine (DA) D2 receptor-mediated GIRK currents (IDA(GIRK)) (IC50: 7.0 μM), with antidepressant-like effec...
T2092 Amitifadine hydrochloride 410074-74-7 98%
Amitifadine hydrochloride
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
T1201 Sulpiride 15676-16-1 98%
Sulpiride
Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.
T6951 Pramipexole dihydrochloride hydrate 191217-81-9 98%
Pramipexole dihydrochloride hydrate
Pramipexole dihydrochloride hydrate (Mirapex) is the hydrochloride salt of pramipexole, a benzothiazole derivative. As a nonergot dopamine agonist, pramipexole b...
T0076 Paliperidone 144598-75-4 98%
Paliperidone
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
T23380 Sonepiprazole 170858-33-0 98%
Sonepiprazole
rat and human dopamine D4 receptor antagonist
T7553 (+)-PD 128907 hydrochloride 300576-59-4 98%
(+)-PD 128907 hydrochloride
(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
T0043 Octodrine 543-82-8 98%
Octodrine
Octodrine (2-Amino-6-methylheptane) is a local anesthetic and vasoconstrictor, but mainly as a pharmaceutical intermediate of Octamylamine.
T60075 Dopamine D2 receptor agonist-2 1610591-93-9 98%
Dopamine D2 receptor agonist-2
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
T12352L Oxidopamine hydrobromide 636-00-0 98%
Oxidopamine hydrobromide
Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
T9827 Carfenazine 2622-30-2 98%
carfenazine
carfenazine targets the Dopamine receptor and is used for schizophrenia research.
Aplindore Fumarate
T30098
Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors,...
Lurasidone hydrochloride
T1735
Lurasidone hydrochloride (Lurasidone HCl) is a thiazole derivative and atypical antipsychotic agent that functions as a dopamine D2 receptor antagonist; serotoni...
BisfluoroModafinil
T4262
CRL-40940 is a selective dopaminergic reuptake inhibitor
DOPEXAMINE
T8653
Dopexamine is a dopaminergic agonist
BP 897 hydrochloride
T14767
BP 897 is a potent and selective agonist of dopamine D3 receptor and it is a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 re...
Fananserin
T15270
Fananserin is an effective, selective and oral active antagonist of 5-HT2 (Ki = 0.37 nM for the rat 5-HT2A). Fananserin is an antagonist of human D4 receptor (Ki...
Levosulpiride
T1211
Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
Minaprine
T0338
Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.
Metoclopramide hydrochloride hydrate
T8385
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction. It...
Tipepidine hydrochloride
T13164
Tipepidine hydrochloride is a reversible inhibitor of dopamine (DA) D2 receptor-mediated GIRK currents (IDA(GIRK)) (IC50: 7.0 μM), with antidepressant-like effec...
Amitifadine hydrochloride
T2092
Amitifadine hydrochloride (EB-1010 hydrochloride) is a triple reuptake inhibitor (TRI) or serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI).
Sulpiride
T1201
Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.
Pramipexole dihydrochloride hydrate
T6951
Pramipexole dihydrochloride hydrate (Mirapex) is the hydrochloride salt of pramipexole, a benzothiazole derivative. As a nonergot dopamine agonist, pramipexole b...
Paliperidone
T0076
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
Sonepiprazole
T23380
rat and human dopamine D4 receptor antagonist
(+)-PD 128907 hydrochloride
T7553
(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Octodrine
T0043
Octodrine (2-Amino-6-methylheptane) is a local anesthetic and vasoconstrictor, but mainly as a pharmaceutical intermediate of Octamylamine.
Dopamine D2 receptor agonist-2
T60075
Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Oxidopamine hydrobromide
T12352L
Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
carfenazine
T9827
carfenazine targets the Dopamine receptor and is used for schizophrenia research.
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TargetMol