Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.

Cat. No.	Product name	CAS No.	Purity
T12928	SK33	1928724-23-5	99.55%
T12928	SK33 is a potent and tissue selective anti-androgen agent. SK33 reduces androgen receptor (AR) transcriptional activity.
T14116	ACP-105	899821-23-9	99.53%
T14116	ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist activity relative to the natural androgen testostero...
T10896L	CSRM617 hydrochloride	1353749-74-2	99.47%
T10896L	CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
T8709	Nandrolone phenylpropionate	62-90-8	99.46%
T8709	Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
T1261	Medroxyprogesterone Acetate	71-58-9	99.45%
T1261	Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective ...
T3137	Boldenone Undecylenate	13103-34-9	99.39%
T3137	Boldenone Undecylenate (Parenabol) is a synthetic steroid.
T26539	AC-262536	870888-46-3	99.38%
T26539	AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
T29111	VPC-13566	218464-59-6	99.37%
T29111	VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the B...
T3618	GSK-2881078	1539314-06-1	99.33%
T3618	GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting t...
T2895	Lupeol	545-47-1	99.31%
T2895	Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
T14008	2,2,5,7,8-Pentamethyl-6-Chromanol	950-99-2	99.3%
T14008	2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol), which has potent androgen receptor (AR) signaling modulation and ...
TCS1372	Atraric acid	4707-47-5	99.27%
TCS1372	Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of pro...
T9246	JNJ-63576253	2110428-64-1	99.27%
T9246	JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
T3357	Clascoterone	19608-29-8	99.26%
T3357	Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.
T16090L	MK-0773 FA		99.17%
T16090L	MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is a selective androgen receptor modulator with an IC50 value of 6.6 nM for AR, which can be used for the prevent...
T8217	Enzalutamide carboxylic acid	1242137-15-0	99.17%
T8217	Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
T10359	AR antagonist 1	1818885-54-9	99.07%
T10359	AR antagonist 1 is a potent antagonist of the androgen receptor. It binds to E3 ligase ligands with weak binding affinities to VHL protein in the synthesis of PR...
T22263	Bavdegalutamide	2222112-77-6	99.04%
T22263	Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR). Bavdegalutamide can be used in studies about prostate cancer. Bavdegalutamide shows ora...
T5100	DJ-V-159	2253744-53-3	99%
T5100	DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member A (GPRC6A).
T6829	EPI-001	227947-06-0	99%
T6829	EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.