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Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .
Cat. No. Product name CAS No. Purity Chemical Structure
T6533 Hexestrol 84-16-2 100%
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
T39710 ARV-471 2229711-68-4 97.15%
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
T2882 Genistin 529-59-9 97.65%
Genistin is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anti...
T15788 LSZ-102 2135600-76-7 97.84%
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
T0301 Ethisterone 434-03-7 97.96%
Ethisterone is a progestogen hormone.
T5S0543 Isocurcumenol 24063-71-6 98%
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
T7299 β-Estradiol 17-acetate 1743-60-8 98%
beta-estradiol 17-acetate is a metabolite of estradiol.
T0035 Dienestrol 84-17-3 98%
Dienestrol is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the vagina and m...
T2544 Bazedoxifene acetate 198481-33-3 98%
Bazedoxifene acetate is a novel selective estrogen receptor modulator (SERM).
T7313 Enclomiphene citrate 7599-79-3 98%
Enclomiphene citrate is a non-steroidal estrogen receptor antagonist,with antioestrogenic property
T1549 Raloxifene hydrochloride 82640-04-8 98%
Raloxifene hydrochloride is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estroge...
T5624 Bisphenol B 77-40-7 98%
Bisphenol B has a binding affinity for estrogen receptors.
T5633 H3B-5942 2052128-15-9 98%
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
T5835 PROTAC ERRα ligand 2 2306388-57-6 98%
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
T5531 GSK-4716 101574-65-6 98%
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
T1571 Estriol 50-27-1 98.05%
Estriol is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen...
T12832 Amcenestrant 2114339-57-8 98.13%
SAR439859 is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER (with an EC50 of 0.2 nM fo...
T15249 Estrogen receptor modulator 1 63676-22-2 98.14%
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active a...
T15364 G-1 881639-98-1 98.14%
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
T20744 Nylestriol 39791-20-3 98.16%
Nylestriol is an agonist of estrogen receptor.
Hexestrol
T6533
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
ARV-471
T39710
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
Genistin
T2882
Genistin is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anti...
LSZ-102
T15788
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
Ethisterone
T0301
Ethisterone is a progestogen hormone.
Isocurcumenol
T5S0543
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
β-Estradiol 17-acetate
T7299
beta-estradiol 17-acetate is a metabolite of estradiol.
Dienestrol
T0035
Dienestrol is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the vagina and m...
Bazedoxifene acetate
T2544
Bazedoxifene acetate is a novel selective estrogen receptor modulator (SERM).
Enclomiphene citrate
T7313
Enclomiphene citrate is a non-steroidal estrogen receptor antagonist,with antioestrogenic property
Raloxifene hydrochloride
T1549
Raloxifene hydrochloride is a second generation selective estrogen receptor modulator (SERM) used to prevent osteoporosis in postmenopausal women. It has estroge...
Bisphenol B
T5624
Bisphenol B has a binding affinity for estrogen receptors.
H3B-5942
T5633
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
PROTAC ERRα ligand 2
T5835
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
GSK-4716
T5531
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
Estriol
T1571
Estriol is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen...
Amcenestrant
T12832
SAR439859 is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER (with an EC50 of 0.2 nM fo...
Estrogen receptor modulator 1
T15249
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active a...
G-1
T15364
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
Nylestriol
T20744
Nylestriol is an agonist of estrogen receptor.
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