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men 1703

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
Dapolsertib
SEL24-B489, SEL 24-B489, MEN1703, MEN 1703
T390851616359-00-2
Dapolsertib (SEL24-B489) is an orally bioavailable and potent PIM and FLT3-ITD inhibitor, inhibiting PIM1, PIM2, and PIM3, decreasing PIM substrate phosphorylation, and inducing dose-dependent apoptosis in leukemia cells.
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7-10 days
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