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Search Result

Search Results for " glutaminase "

Targets

Glutaminase Glutaminase

20

Compounds

1

Natural Products

2

Recombinant Proteins

1

Libraries

Cat No. Product Name Synonyms Targets
T3964 Glutaminase C-IN-1 Compound 968,Glutaminase Inhibitor Compound 968 Glutaminase
Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.
T37385 Glutaminase-IN-3 Glutaminase
Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
T11421 Glutaminase-IN-1 CB839 derivative transporter
Glutaminase-IN-1 (CB839 derivative), a novel 1,3,4-selenodiazepine renal-type glutaminase (KGA) variant inhibitor, showed antitumor activity in an aggressive H22 hepatocellular carcinoma xenograft model.
T78892 Glutaminase C-IN-2 Glutaminase
Glutaminase C-IN-2 (compound 11), an allosteric inhibitor of glutaminase C (GAC), exhibits potent inhibitory activity with an IC50 of 10.64 nM. By disrupting glutamine metabolism, this compound modulates cellular metabol...
T63137 Glutaminase-IN-4
Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).
T83914 Glutaminase C Inhibitor 11
Glutaminase C Inhibitor 11 is a potent inhibitor specifically targeting Glutaminase C (GAC), demonstrating significant inhibition of GAC enzyme activity with an EC50 value of 10.64 nM. It effectively diminishes the viabi...
T6791 BPTES transporter , Glutaminase
BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.
T3968 GK921 Glutaminase
GK921 is a transglutaminase 2 (TGase) inhibitor.
T6797 Telaglenastat CB 839,CB839,CB-839 transporter , Glutaminase , Autophagy
Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.
T20121 L-Albizziin NSC-132089,L-beta-Ureidoalanine,L-Albizziine,Albizzine,NSC 132089,Albizziin Glutaminase
L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.
T78362 Transglutaminase TG
Transglutaminase (TG) is a thiolase that induces intermolecular cross-linking of proteins, by catalysing the formation of isopeptide bonds between the γ-carboxamide group of glutamine residues and the primary ε-amine gro...
T17206 UPGL00004 Others , Glutaminase
UPGL00004 is a potent glutaminase C (GAC) inhibitor with an IC50 of 29 nM. Kd of UPGL00004 for GAC was 27 nM. UPGL00004 has a strong inhibitory effect on the proliferation of highly aggressive triple negative breast canc...
T11412 IPN60090 GLS1-IN-1 Others , transporter
IPN60090 is a novel, potent, orally bioavailable, renal-type glutaminase (GLS1)-specific inhibitor with an IC50 value of 31 nM for GLS1. IPN60090 has potential anticancer and immunostimulant/immunomodulatory activity, se...
T39309 Telaglenastat hydrochloride CB-839 hydrochloride
Telaglenastat (CB-839) hydrochloride is a first-in-class, reversible, and orally active inhibitor of glutaminase 1 (GLS1). It selectively inhibits the splice variants of GLS1, specifically KGA (kidney-type glutaminase) a...
T15613 JHU-083 Others
JHU-083 is a selective glutaminase antagonist. JHU-083 blocks glutaminase activity in brain CD11b+ cells. JHU-083 also experimental cerebral malaria (ECM) resulting in a net decrease of glutamate levels in the animals.
T28961 THDP-17 THDP 17,THDP17
THDP-17 is a inhibitor of glutaminase. THDP-17 shows a partial uncompetitive inhibition in vitro.
T64259 GLS1 Inhibitor-5
GLS1 Inhibitor-5 (compound 24y) is a selective, orally active inhibitor of glutaminase 1 (GLS1) (IC50: 68 nM). gLS1 Inhibitor-5 induces apoptosis and exhibits anti-tumour effects.
T37222 GLS1 Inhibitor
GLS1 inhibitor is an inhibitor of glutaminase 1 (GLS1; IC50= 0.021 μM).1It inhibits the growth of NCI H1703 non-small cell lung cancer (NSCLC) cellsin vitro(GI50= 0.011 μM). GLS1 inhibitor (100 mg/kg) reduces tumor growt...
T39544 IPN60090 dihydrochloride IPN60090 dihydrochloride
IPN-60090 dihydrochloride is a potent and specific inhibitor of glutaminase 1 (GLS1) with a remarkable inhibition constant (IC50) of 31 nM. It does not exhibit any inhibitory activity against GLS-2. Furthermore, IPN-6009...
T73458 LWG-301
LWG-301, an allosteric inhibitor of Glutaminase 1 (GLS1), demonstrates a potent inhibition with an IC50 value of 7 nM. It effectively impedes glutamine metabolism and elevates intracellular ROS levels, thereby inducing a...
Cat No. Product Name Synonyms Targets
T8373 6-Diazo-5-oxo-L-nor-Leucine DON,L-6-Diazo-5-oxonorleucine,Diazooxonorleucine Influenza Virus , Glutaminase , Antibacterial , Antibiotic
6-Diazo-5-oxo-L-nor-Leucine (L-6-Diazo-5-oxonorleucine) is an antagonist of glutaminases (Ki : 6 μM). It is an antineoplastic antibiotic produced by an unidentified species of Streptomyces from Peruvian soil.

Natural Products

6-Diazo-5-oxo-L-nor-Leucine
T8373
Synonym: DON,L-6-Diazo-5-oxonorleucine,Diazooxonorleucine
Target: Influenza Virus, Glutaminase, Antibacterial, Antibiotic

Recombinant Proteins

Species：
Human (2)
Expression System：
Baculovirus-Insect Cells (2)
Tag：
His (2)
Cat No. Product Name Species Expression System
TMPY-01355 Transglutaminase 2/TGM2 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Protein-glutamine gamma-glutamyltransferase 2, also known as Tissue transglutaminase, Transglutaminase C, Transglutaminase-2, and TGM2, is a member of the transglutaminase superfamily. TGM2 plays a role in cell growth an...
TMPY-02129 Transglutaminase 3/TGM3 Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
Transglutaminases (TGase) are a family of calcium-dependent acyl-transfer enzymes ubiquitously expressed in mammalian cells and responsible for catalyzing covalent cross-links between proteins or peptides. Transglutamina...
Cat No. Product Name
L2550 Glutamine Metabolism Compound Library

580 compounds
A unique collection of 580 glutamine metabolism related compounds can be used for high throughput screening (HTS) and high content screening (HCS), and also is an effective tool for research in glutamine metabolism and ...

Libraries

Glutamine Metabolism Compound Library
L2550
Compounds: 580
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