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Search Results for " sstr "

19

Compounds

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T76544 Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .
T9692 Paltusotine Somatostatin
Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients
TP2207 Pasireotide Acetate Somatostatin
Pasireotide Acetate is a stable cyclohexapeptide somatostatin mimic
T2584 Octreotide SMS 201-995 Somatostatin
Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.
T4119 Octreotide Acetate SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate) Somatostatin
Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.
T13022 SSTR5 antagonist 2 Others
SSTR5 antagonist 2 is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5),with potential to treat type 2 diabetes mellitus (T2DM).
T13005 SSTR5 antagonist 1 Others
SSTR5 antagonist 1 is a selective, and orally available antagonist of somatostatin receptor subtype 5 (SSTR5)(IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively).
T13022L SSTR5 antagonist 2 TFA Others
SSTR5 antagonist 2 TFA is a highly potent, oral active and selective antagonist of somatostatin (receptor) subtype 5 (SSTR5), with potential to treat type 2 diabetes mellitus (T2DM).
TP2045 CH 275
Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin r...
T61130 SSTR4 agonist 3
SSTR4 agonist 3 is a potent compound that activates the SSTR4 receptor. The SSTR4 receptor is highly expressed in the hippocampus and neocortex, which are regions associated with memory, learning, and Alzheimer's disease...
T60911 SSTR4 agonist 4
SSTR4 agonist 4 is a potent SSTR4 agonist that has the potential for the pain research. SSTR4 agonists are effective in rodent models of pain associated with acute and chronic associated anti-peripheral nociceptive and a...
T64119 SSTR5 antagonist 2 hydrochloride
SSTR5 antagonist 2 hydrochloride is a potent, orally active, selective growth hormone inhibitory hormone (receptor) subtype 5 (SSTR5) antagonist that has shown potential for investigation in type 2 diabetes.
T60784 SSTR4 agonist 2
SSTR4 agonist 2 is a potent somatostatin receptor subtype 4 (SSTR4) agonist that has the potential in SSTR4-related medical disorders research. SSTR4 pathway inhibits the processes of nociceptive and inflammatory [1].
T80238 NODAGA-LM3 TFA
NODAGA-LM3 TFA, a SSTR2 antagonist, can be radiolabeled with ^68Ga for PET imaging applications, particularly in the visualization of SSTR-positive paragangliomas [1] [2].
T80237 NODAGA-LM3
NODAGA-LM3, when labeled with ^68Ga, serves as a PET imaging agent. As an SSTR2 antagonist, ^68Ga-NODAGA-LM3 is utilized for the visualization of SSTR-positive paragangliomas [1] [2].
T76980 Tidutamab
Tidutamab (XmAb-18087) is a humanized and affinity-optimized bispecific antibody (bsAb) targeting SSTR2 binding domain and T-cell binding domain (CD3) . Tidutamab possesses a full Fc domain to maintain long serum half-li...
T78110 DOTA-LM3 TFA
DOTA-LM3 TFA is a somatostatin receptor (SSTR) antagonist with the molecular structure p-Cl-Phe-cyclo(D-Cys-Tyr-D-4-amino-Phe(carbamoyl)-Lys-Thr-Cys)D-Tyr-NH2. It is effectively used in tracing tumors in vivo through iso...
T80155 DOTA-LM3
DOTA-LM3 is a somatostatin receptor (SSTR) antagonist, with LM3 denoting the peptide sequence p-Cl-Phe-cyclo(D-Cys-Tyr-D-4-amino-Phe(carbamoyl)-Lys-Thr-Cys)D-Tyr-NH2. It is utilized in the isotopic labeling of tumors for...
T37109 BIM-23190 hydrochloride
BIM-23190 hydrochloride, a somatostatin analog, a selective SSRT2 and SSRT5 agonist, exhibits Ki values of 0.34 nM and 11.1 nM for SSTR2 and SSTR5, respectively. BIM-23190 can be used in the study for cancer and acromega...

Recombinant Proteins

Cat No. Product Name Species Expression System
TMPY-06360 SSTR2/SSTR2B Protein-VLP, Human, Recombinant Human HEK293
TMPY-00374 SSTR1 Protein, Human, Recombinant (hFc) Human HEK293
TMPY-06364 SSTR2/SSTR2A Protein-VLP, Human, Recombinant Human HEK293
TargetMol