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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8596 | Ceefourin 1 | MRP | |
Ceefourin 1 is a highly selective multidrug resistance protein 4 (MRP4) inhibitor. | |||
T3148 | MK-571 sodium | L-660711 (sodium salt),L-660711 sodium salt,Verlukast sodium,L-660711,MK571,MK-571 sodium salt,Propanoic acid | Leukotriene Receptor , LTR |
MK-571 sodium (L-660711 sodium salt) is a selective, orally active antagonist of the CysLT1 receptor. MK-571 sodium is a multidrug resistance protein-2 (ABCC2, Mrp2) inhibitor used to demonstrate the role of Mrp2 in the ... | |||
T17072 | Thiethylperazine dimaleate | Toresten,Thiethylperazine maleate,Norzine | Dopamine Receptor , Antibacterial , ABC , Histamine Receptor |
Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 and possesses antimicrobial, anti-emetic, and antipsychotic e... | |||
T11071 | Dofequidar fumarate | MS-209 | P-gp |
Dofequidar fumarate (MS-209)(MS-209 fumarate), a quinoline-based compound administered orally, is known for counteracting multidrug resistance (MDR) through the inhibition of ABCB1/P-glycoprotein (P-gp) and ABCC1/MDR-ass... | |||
T61915 | Thiethylperazine | ||
Thiethylperazine is a phenothiazine derivative. Thiethylperazine is a histamine H1 receptor and dopamine D2 receptor antagonist with oral activity. Thiethylperazine is also a selective ABCC1 activator, which can reduce a... |
Cat No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-01711 | ABCC1 Protein, Human, Recombinant (His) | Human | E. coli |
Mediates export of organic anions and drugs from the cytoplasm. Mediates ATP-dependent transport of glutathione and glutathione conjugates, leukotriene C4, estradiol-17-beta-o-glucuronide, methotrexate, antiviral drugs a... |