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Cat No. | Product Name | Synonyms | Targets |
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T6240 | Palbociclib Isethionate | Palbociclib (PD0332991) Isethionate,PD 0332991 isethionate | CDK |
Palbociclib Isethionate (PD 0332991 isethionate) is a selective inhibitor of CDK4/6 (IC50s: 11/16 nM). It exhibits no inhibition against a panel of 36 additional protein kinases. | |||
T1654 | Pentamidine isethionate | Pentamidine isethionate salt,Pentamidine diisethionate | Phosphatase , Antibacterial , Antibiotic , Parasite , Antifungal |
Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent. | |||
T68657 | Asulacrine isethionate | ||
Asulacrine isethionate (CI-921) is a topoisomerase ll inhibitor with antineoplastic properties. Asulacrine blocks DNA replication and RNA and protein synthesis. | |||
T29977 | Amicarbalide diisethionate | ||
Amicarbalide diisethionate is a bioactive chemical. | |||
T36482 | Lamotrigine isethionate | ||
Water-soluble salt of lamotrigine . Displays anticonvulsant effects and inhibits glutamate release, possibly through inhibition of Na+, K+ and Ca2+ currents. Leach et al (1991) Neurochemical and behavioral aspects of lam... | |||
T32279 | JB-11 isethionate | NSC328564,NSC-328564,NSC 328564 | |
JB-11 isethionate is a bioactive chemical. | |||
T28048 | Mivobulin Isethionate | NSC-613863,CI-980,NSC-635370,NSC-613862,NSC-350386 | |
Mivobulin is a tubulin inhibitor potentially for the treatment of glioma, malignant melanoma, prostate, ovarian cancer. CI-980 acts at the colchicine-binding site. | |||
T34144 | Propamidine isethionate | ||
Propamidine isethionate is a biaoctive chemical. | |||
T68684 | Piritrexim isethionate | ||
Piritrexim isethionate is a lipid-soluble inhibitor of dihydrofolate reductase (DHFR) that appears to be an active agent in patients with metastatic urothelial cancer when administered as a 5-day, low-dose oral schedule. |
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1085 | L-Glutathione reduced | GSH,Isethion,Glutathione,γ-L-Glutamyl-L-cysteinyl-glycine,Glutathion,Tathion | Ferroptosis , Reactive Oxygen Species , Endogenous Metabolite , Glutathione reductase |
L-Glutathione reduced (Glutathione) is a tripeptide with many roles in cells. It conjugates to drugs to make them more soluble for excretion, is a cofactor for some enzymes, is involved in protein disulfide bond rearrang... | |||
T5303 | Isethionic acid sodium salt | Sodium isethionate | Others , Endogenous Metabolite |
Isethionic acid sodium salt (Sodium isethionate) is an organosulfur compound containing a short chain alkane sulfonate linked to a hydroxyl group. Mammals are able to endogenously synthesize Isethionic acid sodium salt v... | |||
T20854 | Isethionic acid | Hydroxyethylsulfonic acid,Ethanolsulfonic acid | |
Isethionic acid, a major metabolite in F. cylindrus, is an organosulfur compound containing a short-chain alkane sulfonate linked to a hydroxyl group. It is a water-soluble liquid for the manufacture of mild, biodegradab... |