TQ0159 |
U-73343
|
142878-12-4
|
99.06%
|
|
U-73343 is an inactive analog of U-73122 and can be used as a negative control. It dose-dependently inhibits acid secretion irrespective of the stimulant. It is ...
|
T11149 |
Ecopladib
|
381683-92-7
|
99.02%
|
|
Ecopladib (PLA 725) is a sub-micromolar inhibitor of cytosolic phospholipase A2α (cPLA2α), with IC50s of 0.15 μM and 0.11 μM in the GLU micelle and rat whole blo...
|
T21606L |
Anti-Inflammatory Peptide 1 Acetate
|
T21606L
|
98.95%
|
|
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) possesses a potent anti-inflammatory activity in vivo and is a strong inhibitor of phospholipase A2 (PLA2), ...
|
T4192 |
Hnps-PLA Inhibitor
|
185298-58-2
|
98.95%
|
|
Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
|
T4511 |
ST271
|
106392-48-7
|
98.94%
|
|
ST271 is an effective protein tyrosine kinase (PTK) inhibitor.
|
T60967 |
Atg4B-IN-2
|
2765008-88-4
|
98.86%
|
|
Atg4B-IN-2 is a potent and selective Atg4B inhibitor with anticancer activity that inhibits the activity of Atg4B and PLA2.Atg4B-IN-2 resists the anticancer acti...
|
T60043 |
DPTIP
|
351353-48-5
|
98.80%
|
|
DPTIP is an effective inhibitor of neutral sphingomyelinase 2 with an IC50 value of 30 nM.
|
T2907 |
Tanshinone I
|
568-73-0
|
98.58%
|
|
Tanshinone I (Tanshinone A), an active principle isolated from the herbal medicine Salvia miltiorrhiza, displays cytotoxicity against tumor cells.
|
T4019 |
Cambinol
|
14513-15-6
|
98.47%
|
|
Cambinol (SIRT1/2 Inhibitor IV) is a cell-permeable b-naphthol compound that inhibits the NAD-dependent deacetylase activity of SIRT1/2 (IC50: 56/59 μM, respecti...
|
TP1299 |
Melittin
|
20449-79-0
|
98.37%
|
|
Melittin, a small protein containing 26 amino acid residues, is the principal toxic component of bee venom. Melittin is a PLA2 activator, stimulates the activity...
|
T21651 |
Lansoprazole sodium
|
226904-00-3
|
98.35%
|
|
Lansoprazole sodium (Lansoprazole (sodium)) is a proton pump inhibitor (PPI) and a potent inhibitor of gastric acidity which is widely used in the therapy of gas...
|
T17239 |
VU0155069
|
1130067-06-9
|
98.32%
|
|
VU0155069 strongly inhibits the invasive migration of several cancer cell lines in transwell assays. VU0155069 is a selective phospholipase D1 inhibitor (IC50: 4...
|
T13632 |
D-Erythro-dihydrosphingosine
|
764-22-7
|
98.03%
|
|
D-Erythro-dihydrosphingosine (C18-Dihydrosphingosine) inhibits arachidonic acid release and cPLA2α activity.
|
T8236 |
RHC 80267
|
83654-05-1
|
98%
|
|
RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)
|
T2044 |
Varespladib
|
172732-68-2
|
98%
|
|
Varespladib (LY315920), a specific and effective human non-pancreatic secretory phospholipase A2 (hnsPLA) inhibitor(IC50=7 nM), has been investigated for the tre...
|
T7280 |
CAY10594
|
1130067-34-3
|
98%
|
|
CAY10594 is a potent phospholipase D2(PLD2) inhibitor. CAY10594 ameliorates acetaminophen-induced acute liver injury by regulating the phosphorylated-GSK-3β/JNK ...
|
T2282 |
RPI-1
|
269730-03-2
|
98%
|
|
RPI-1 is a competitive, potent ATP-dependent Ret kinase inhibitor.
|
T6243 |
U-73122
|
112648-68-7
|
97.98%
|
|
U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.
|
T70955 |
Vinaxanthone
|
133293-89-7
|
97.65%
|
|
Vinaxanthone (SM-345431) is a small molecule compound derived from Penicillium chrysogenum that is a selective and potent semaphorin3A, phospholipase C (PLC), an...
|
T0757 |
Omeprazole
|
73590-58-6
|
97.61%
|
|
Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor (exosome inhibito...
|