T0979 |
Dequalinium chloride
|
522-51-0
|
99.58%
|
|
Dequalinium Chloride, a topical bacteriostat, is a selective blocker of apamin-sensitive K+ channels. It is used in wound dressings and mouth infections and may ...
|
T6139L |
A-674563 2HCl(552325-73-2(fb-2hcl))
|
T6139L
|
99.57%
|
|
A-674563 2HCl is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.
|
T3211 |
Midostaurin
|
120685-11-2
|
99.56%
|
|
PKC412(Midostaurin; CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor. Midostaurin inhibits protein kinase C alpha (PKCalpha), vascular endothelia...
|
T7792 |
Hispidin
|
555-55-5
|
99.55%
|
|
Hispidin is a polyphenol originally, including antioxidant, anti-inflammatory, and cytoprotective properties
|
T0033 |
Miltefosine
|
58066-85-6
|
99.51%
|
|
Miltefosine is the treatment of visceral and cutaneous leishmaniasis drug , and is proceeding clinical trials for this in several countries. Several medical agen...
|
T6S0923 |
Hypericin
|
548-04-9
|
99.51%
|
|
1. Hypericin has antineoplastic activity. 2. Hypericin has antibiotic and antiviral activities. 3. Hypericin has antidepressive activity through inhibiting monoa...
|
T13314 |
VTX-27
|
1321924-70-2
|
99.49%
|
|
VTX-27 is a selective inhibitor of protein kinase C θ (PKC θ) (Kis: 0.08 nM and 16 nM for PKC θ and PKC δ).
|
T13384L |
Y-33075 dihydrochloride
|
173897-44-4
|
99.43%
|
|
Y-33075 dihydrochloride is a selective inhibitor of ROCK(IC50 of 3.6 nM).
|
T0610 |
Piceatannol
|
10083-24-6
|
99.39%
|
|
Piceatannol is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine kinases and inhibits NF-κB activat...
|
T5796 |
Plantainoside D
|
147331-98-4
|
99.39%
|
|
Plantainoside D shows potent antioxidative effects as those of ascorbic acid, it shows angiotensin-converting enzyme (ACE) inhibitory inhibitory activity in vitr...
|
T12148 |
N-Desmethyltamoxifen hydrochloride
|
15917-65-4
|
99.34%
|
|
N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.
|
TN1136 |
Procyanidin A1
|
103883-03-0
|
99.23%
|
|
Procyanidin A1 (Proanthocyanidin A1) has antiallergic effects, it inhibits degranulation downstream of protein kinase C activation or Ca2+; influx from an intern...
|
T6643 |
Ro 31-8220 Mesylate
|
138489-18-6
|
99.18%
|
|
Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor for PKC-α/βI/βII/γ/ε (IC50: 5/24/14/27/24 nM), and also shows potent inhibition agai...
|
T6932 |
PD168393
|
194423-15-9
|
99.13%
|
|
PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, FGFR, PDGFR, and insulin.
|
TN1047 |
Ingenol mebutate
|
75567-37-2
|
99.04%
|
|
Ingenol mebutate is a potent activator of PKC subtypes including PKC-α, PKC-β, PKC-γ, PKC-δ, and PKC-ε with Kis of 0.3, 0.105, 0.162, 0.376, and 0.171 nM. Ingeno...
|
T27525 |
HA-1004
|
91742-10-8
|
99.03%
|
|
HA-1004 is a inhibitor of PKG, PKA, PKC and MLC.
|
T10549 |
Bisindolylmaleimide VIII acetate
|
138516-31-1
|
99%
|
|
Bisindolylmaleimide VIII acetate is a potent and selective PKC inhibitor (IC50: 158 nM for rat brain PKC). It has IC50s of 53, 195, 163, 213, and 175 nM for PKC-...
|
T2S0531 |
Pinoresinol dimethyl ether
|
29106-36-3
|
98.98%
|
|
Pinoresinol dimethyl ether is a natural product for research related to life sciences. The catalog number is T2S0531 and the CAS number is 29106-36-3.
|
T35827L |
PKCε Inhibitor Peptide acetate
|
|
98.93%
|
|
PKCε Inhibitor Peptide acetate is a selective PKCε inhibitor containing the site for its specific receptor for activated C kinase (RACK). PKCε Inhibitor Peptide ...
|
TN1299 |
Desmethylglycitein
|
17817-31-1
|
98.93%
|
|
6,7,4'-Trihydroxyisoflavone, is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which has antioxidant, and anti-cancer acti...
|