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PKC

Protein kinase C, commonly abbreviated to PKC, is a family of protein kinase enzymes that are involved in controlling the function of other proteins through the phosphorylation of hydroxyl groups of serine and threonine amino acid residues on these proteins, or a member of this family. PKC enzymes in turn are activated by signals such as increases in the concentration of diacylglycerol (DAG) or calcium ions (Ca2+). Hence PKC enzymes play important roles in several signal transduction cascades.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T5423 PKC-theta inhibitor 736048-65-0
PKC-theta inhibitor
PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.
T12496 PKC-theta inhibitor 1 1160501-81-4 98%
PKC-theta inhibitor 1
PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)
TN1542 Cycloheterophyllin 36545-53-6 98%
Cycloheterophyllin
Cycloheterophyllin has an antioxidant effect, it is a photoprotective agent that inhibits ultraviolet A (UVA)-induced oxidative stress and damage, and could be u...
T13637 DCP-LA 28399-31-7 98%
DCP-LA
DCP-LA (FR236924), linoleic acid derivatives, selective and direct activation of PKCε.
T78220 SAMβA TFA 98%
SAMβA TFA
SAMβA TFA, a selective antagonist of Mfn1-βIIPKC association conjugated to the cell permeable peptide TAT47-57, is a rationally designed inhibitor that improves ...
T78833 AJH-836 388621-67-8 98%
AJH-836
AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) of 4.5 nM for PKCα, and facilitates the translocation of Mu...
T79493 HIV-1 protease-IN-10 98%
HIV-1 protease-IN-10
HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM) and demo...
T80070 PKCβII Peptide Inhibitor I 862502-26-9 98%
PKCβII Peptide Inhibitor I
PKCβII Peptide Inhibitor I, a specific PKCβII inhibitor, exhibits cardioprotective properties in a rat cardiac ischemia/reperfusion injury model and mitigates va...
T80248 PKCε (85-92) 207111-98-6 98%
PKCε (85-92)
PKCε (85-92) is a biologically active peptide that functions as a specific activator of ε-PKC and induces MARCKS phosphorylation in wild-type cells, but does not...
T80249 Epsilon-V1-2, Cys-conjugated 98%
Epsilon-V1-2, Cys-conjugated
Epsilon-V1-2, a Cys-conjugated, is a biologically active peptide known as the εPKC-specific inhibitor. It hampers εPKC functionality by obstructing its transloca...
T80504 ɛPKC(85–92),Myristoylated 1072301-79-1 98%
ɛPKC(85–92),Myristoylated
Myristoylated ?PKC(85–92) is a myristic acid-conjugated, cell-permeable peptide activator of PKC? that has been shown to increase nitric oxide (NO) release in cu...
T80505 PKCα (C2-4) inhibitor peptide 98%
PKCα (C2-4) inhibitor peptide
PKCα (C2-4) inhibitor peptide is a specific antagonist to PKCα that impedes the α1A-adrenoreceptor agonist A-61603 [1] from inhibiting I_Kr.
T80507 PKCθ pseudosubstrate peptide inhibitor,myristoylated 98%
PKCθ pseudosubstrate peptide inhibitor,myristoylated
Myristoylated PKCθ pseudosubstrate peptide inhibitor is a synthetic peptide utilized to investigate the mechanism of action of protein kinase C theta (PKCθ) [1]....
T80508 PKCη pseudosubstrate inhibitor,myristoylated 908012-19-1 98%
PKCη pseudosubstrate inhibitor,myristoylated
Myristoylated PKCη pseudosubstrate inhibitor is a cell-permeable compound utilized to investigate the mechanism of action of PKCη [1].
T80509 PKC 20-28,myristoylated 98%
PKC 20-28,myristoylated
Myristoylated protein kinase C inhibitor 20-28 (PKC 20-28,myristoylated) is a cell-permeable inhibitor of protein kinase C, utilized in cancer research [1].
T80511 PKCε inhibitor peptide,myristoylated 98%
PKCε inhibitor peptide,myristoylated
Myristoylated PKCε inhibitor peptide (Myr-PKCε-) is a cell-permeable inhibitor consisting of a peptide linked to myristic acid that specifically inhibits protein...
T80514 TAT-SAMβA 98%
TAT-SAMβA
TAT-SAMβA, an RNAENFDRF (SAMβA) peptide conjugated to the TAT 47–57 protein-derived cell-penetrating peptide, acts as a selective antagonist of the Mfn1-βIIPKC a...
T80550 N-myristoyl-RKRTLRRL 152246-40-7 98%
N-myristoyl-RKRTLRRL
N-myristoyl-RKRTLRRL is a compound that impedes the binding of protein kinase C (PKC) substrates and inhibits calcium (Ca2+)- and phosphatidylserine (PS)-depende...
T81449 PKC-ε translocation inhibitor peptide 98%
PKC-ε translocation inhibitor peptide
PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαR tra...
T12494 PKC-IN-1 1046787-18-1 98%
PKC-IN-1
PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6, 2...
PKC-theta inhibitor
T5423
PKC-theta inhibitor is PKC-θinhibitor, with an IC50 of 12 nM.
PKC-theta inhibitor 1
T12496
PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)
Cycloheterophyllin
TN1542
Cycloheterophyllin has an antioxidant effect, it is a photoprotective agent that inhibits ultraviolet A (UVA)-induced oxidative stress and damage, and could be u...
DCP-LA
T13637
DCP-LA (FR236924), linoleic acid derivatives, selective and direct activation of PKCε.
SAMβA TFA
T78220
SAMβA TFA, a selective antagonist of Mfn1-βIIPKC association conjugated to the cell permeable peptide TAT47-57, is a rationally designed inhibitor that improves ...
AJH-836
T78833
AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) of 4.5 nM for PKCα, and facilitates the translocation of Mu...
HIV-1 protease-IN-10
T79493
HIV-1 protease-IN-10 (Compound 2), exhibiting HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM) and demo...
PKCβII Peptide Inhibitor I
T80070
PKCβII Peptide Inhibitor I, a specific PKCβII inhibitor, exhibits cardioprotective properties in a rat cardiac ischemia/reperfusion injury model and mitigates va...
PKCε (85-92)
T80248
PKCε (85-92) is a biologically active peptide that functions as a specific activator of ε-PKC and induces MARCKS phosphorylation in wild-type cells, but does not...
Epsilon-V1-2, Cys-conjugated
T80249
Epsilon-V1-2, a Cys-conjugated, is a biologically active peptide known as the εPKC-specific inhibitor. It hampers εPKC functionality by obstructing its transloca...
ɛPKC(85–92),Myristoylated
T80504
Myristoylated ?PKC(85–92) is a myristic acid-conjugated, cell-permeable peptide activator of PKC? that has been shown to increase nitric oxide (NO) release in cu...
PKCα (C2-4) inhibitor peptide
T80505
PKCα (C2-4) inhibitor peptide is a specific antagonist to PKCα that impedes the α1A-adrenoreceptor agonist A-61603 [1] from inhibiting I_Kr.
PKCθ pseudosubstrate peptide inhibitor,myristoylated
T80507
Myristoylated PKCθ pseudosubstrate peptide inhibitor is a synthetic peptide utilized to investigate the mechanism of action of protein kinase C theta (PKCθ) [1]....
PKCη pseudosubstrate inhibitor,myristoylated
T80508
Myristoylated PKCη pseudosubstrate inhibitor is a cell-permeable compound utilized to investigate the mechanism of action of PKCη [1].
PKC 20-28,myristoylated
T80509
Myristoylated protein kinase C inhibitor 20-28 (PKC 20-28,myristoylated) is a cell-permeable inhibitor of protein kinase C, utilized in cancer research [1].
PKCε inhibitor peptide,myristoylated
T80511
Myristoylated PKCε inhibitor peptide (Myr-PKCε-) is a cell-permeable inhibitor consisting of a peptide linked to myristic acid that specifically inhibits protein...
TAT-SAMβA
T80514
TAT-SAMβA, an RNAENFDRF (SAMβA) peptide conjugated to the TAT 47–57 protein-derived cell-penetrating peptide, acts as a selective antagonist of the Mfn1-βIIPKC a...
N-myristoyl-RKRTLRRL
T80550
N-myristoyl-RKRTLRRL is a compound that impedes the binding of protein kinase C (PKC) substrates and inhibits calcium (Ca2+)- and phosphatidylserine (PS)-depende...
PKC-ε translocation inhibitor peptide
T81449
PKC-ε Translocation Inhibitor Peptide is a selective modulator that controls the FcγR-mediated internalization rate of opsonized beads without affecting FcαR tra...
PKC-IN-1
T12494
PKC-IN-1 is an ATP-competitive and reversible conventional PKC enzymes inhibitor (PKCα, PKCβI, PKCβII, PKCθ, PKCγ, PKC mu and PKCε with IC50s of 2.3, 8.1, 7.6, 2...
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TargetMol