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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T4196 Betahistine EP Impurity C 5452-87-9 98%
Betahistine EP Impurity C
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
T4195 Betahistine 5638-76-6 97.92%
Betahistine
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but m...
T13352 Wy 49051 113418-56-7 97.9%
Wy 49051
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
T19443 N-Acetylhistamine 673-49-4 97.72%
N-Acetylhistamine
N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.
T79499 KSK68 2566715-91-9 97.22%
KSK68
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 recept...
T3979 Emedastine 87233-61-2 97.1%
Emedastine
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blo...
T0076 Paliperidone 144598-75-4 96.98%
Paliperidone
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
T13566 Bamirastine 215529-47-8 96.68%
Bamirastine
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on alle...
T0965 Histamine 51-45-6 96.63%
Histamine
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial s...
T68122L Oxmetidine FA 96.48%
Oxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
TQ0046 Bavisant 929622-08-2 96.06%
Bavisant
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefu...
T0445L Promethazine hydrochloride 58-33-3 95.36%
Promethazine hydrochloride
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mA...
T40652 Meclizine 569-65-3 95.16%
Meclizine
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptors ...
T16280 Nedocromil 69049-73-6 95%
Nedocromil
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
T0185 Escitalopram 128196-01-0 94.62%
Escitalopram
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
T29096L Vapitadine 793655-64-8 100%
Vapitadine
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
T12054L MK-0249 FA 100%
MK-0249 FA
MK-0249 FA is an orally active, selective and potent histamine H3 inverse agonist for the study of attention deficit, hyperactivity disorder neurodivergent and c...
T61213 PF-03654764 935840-35-0 100%
PF-03654764
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist that inhibits human H3 and rat H3 with Ki values of 1.2 nM and 7.9 nM, re...
T6535 Histamine Phosphate 51-74-1 100%
Histamine Phosphate
Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.
T1470L Fexofenadine hydrochloride 138452-21-8 100%
Fexofenadine hydrochloride
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic...
Betahistine EP Impurity C
T4196
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
Betahistine
T4195
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but m...
Wy 49051
T13352
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
N-Acetylhistamine
T19443
N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.
KSK68
T79499
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 recept...
Emedastine
T3979
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blo...
Paliperidone
T0076
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
Bamirastine
T13566
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on alle...
Histamine
T0965
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial s...
Oxmetidine FA
T68122L
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
Bavisant
TQ0046
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefu...
Promethazine hydrochloride
T0445L
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mA...
Meclizine
T40652
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptors ...
Nedocromil
T16280
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
Escitalopram
T0185
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
Vapitadine
T29096L
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
MK-0249 FA
T12054L
MK-0249 FA is an orally active, selective and potent histamine H3 inverse agonist for the study of attention deficit, hyperactivity disorder neurodivergent and c...
PF-03654764
T61213
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist that inhibits human H3 and rat H3 with Ki values of 1.2 nM and 7.9 nM, re...
Histamine Phosphate
T6535
Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.
Fexofenadine hydrochloride
T1470L
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic...
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TargetMol