T4196 |
Betahistine EP Impurity C
|
5452-87-9
|
98%
|
|
Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.
|
T4195 |
Betahistine
|
5638-76-6
|
97.92%
|
|
Betahistine (Vasomotal) is a histamine analog and H1 receptor agonist that serves as a vasodilator. It is used in MENIERE DISEASE and in vascular headaches but m...
|
T13352 |
Wy 49051
|
113418-56-7
|
97.9%
|
|
Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
|
T19443 |
N-Acetylhistamine
|
673-49-4
|
97.72%
|
|
N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.
|
T79499 |
KSK68
|
2566715-91-9
|
97.22%
|
|
KSK68 is a potent dual sigma-1 and histamine H3 receptor antagonist with potential analgesic activity and high affinity for H3 receptors, sigma-1, sigma-2 recept...
|
T3979 |
Emedastine
|
87233-61-2
|
97.1%
|
|
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity. Emedastine reversibly and competitively blo...
|
T0076 |
Paliperidone
|
144598-75-4
|
96.98%
|
|
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically,...
|
T13566 |
Bamirastine
|
215529-47-8
|
96.68%
|
|
Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on alle...
|
T0965 |
Histamine
|
51-45-6
|
96.63%
|
|
Histamine (Ergamine) is an amine derived by enzymatic decarboxylation of HISTIDINE. It is a powerful stimulant of gastric secretion, a constrictor of bronchial s...
|
T68122L |
Oxmetidine FA
|
|
96.48%
|
|
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
|
TQ0046 |
Bavisant
|
929622-08-2
|
96.06%
|
|
Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist. Bavisant can be used in research on mechanisms of action, involving wakefu...
|
T0445L |
Promethazine hydrochloride
|
58-33-3
|
95.36%
|
|
Promethazine hydrochloride (Promethazine HCl) , the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mA...
|
T40652 |
Meclizine
|
569-65-3
|
95.16%
|
|
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that inhibits the interaction of histamine at H1 receptors ...
|
T16280 |
Nedocromil
|
69049-73-6
|
95%
|
|
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
|
T0185 |
Escitalopram
|
128196-01-0
|
94.62%
|
|
Escitalopram (Seroplex) is a furancarbonitrile that is one of the SEROTONIN UPTAKE INHIBITORS used as an antidepressant. The drug is also effective in reducing e...
|
T29096L |
Vapitadine
|
793655-64-8
|
100%
|
|
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
|
T12054L |
MK-0249 FA
|
|
100%
|
|
MK-0249 FA is an orally active, selective and potent histamine H3 inverse agonist for the study of attention deficit, hyperactivity disorder neurodivergent and c...
|
T61213 |
PF-03654764
|
935840-35-0
|
100%
|
|
PF-03654764 is an orally active, potent, and selective histamine H3 receptor antagonist that inhibits human H3 and rat H3 with Ki values of 1.2 nM and 7.9 nM, re...
|
T6535 |
Histamine Phosphate
|
51-74-1
|
100%
|
|
Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.
|
T1470L |
Fexofenadine hydrochloride
|
138452-21-8
|
100%
|
|
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic...
|