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target/HIV_Protease/4

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    21
    TargetMol | Activity
  • Peptide Products
    6
    TargetMol | inventory
Protease-Activated Receptor-4 diTFA
T7740
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
  • $33
In Stock
Size
QTY
TargetMol | Inhibitor Sale
HIV-1 protease-IN-9
T792952925381-27-5
HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a half-maximal inhibitory concentration (IC_50) of 66.8 nM [1].
  • $1,370
8-10 weeks
Size
QTY
HIV-1 protease-IN-11
T795362925287-54-1
HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacy against a drug-resistant variant [1].
  • $1,970
8-10 weeks
Size
QTY
HIV-1 protease-IN-7
T749422916441-36-4
HIV-1 protease-IN-7 (compound 16) is an orally active HIV-1 protease inhibitor with an IC50 of 3.52 nM and an EC50 of 37 nM [1].
  • Inquiry Price
8-10 weeks
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Protease-Activated Receptor-4
T7380245443-52-1
Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
    7-10 days
    Inquiry
    HIV Protease Substrate 1 TFA
    T76074
    HIV Protease Substrate 1 TFA, a fluorogenic substrate for HIV protease, facilitates the investigation of the enzyme's activity [1].
    • Inquiry Price
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    QTY
    HIV-1, HIV-2 Protease Substrate
    T76502149639-49-6
    HIV-1, HIV-2 Protease Substrate serves as a substrate for the proteases of both HIV-1 and HIV-2, featuring four residues that permit conservative substitutions at the enzyme substrate binding sites [1].
    • Inquiry Price
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    HIV-1 protease-IN-12
    T795372925287-59-6
    HIV-1 protease-IN-12 (compound 35b) is a potent HIV-1 protease inhibitor with an IC50 value of 0.51 nM, demonstrating efficacy against drug-resistant variants [1].
    • $1,970
    8-10 weeks
    Size
    QTY
    HIV-1 integrase inhibitor 4
    T115681638504-66-1
    HIV-1 integrase inhibitor 4 is an HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM.
    • $1,670
    6-8 weeks
    Size
    QTY
    HIV protease-IN-1
    T749392511547-82-1
    HIV protease-IN-1 (compound 1·succinate), a potent non-peptidic inhibitor of HIV protease, is used in AIDS research [1].
    • Inquiry Price
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    HIV Protease Substrate 1
    T39729223769-59-3
    HIV Protease Substrate 1 is a fluorogenic compound that offers insights into the enzymatic activity of HIV protease, making it a valuable tool for studying this aspect.
    • $1,520
    Backorder
    Size
    QTY
    HIV-1 protease-IN-5
    T641122525173-96-8
    HIV-1 protease-IN-5 is an HIV-1 protease inhibitor (IC50: 1.64 nM). HIV-1 protease-IN-5 exhibits significant effects on wild-type and DRV-resistant HIV-1.
    • $1,520
    6-8 weeks
    Size
    QTY
    HIV-1 protease-IN-1
    T634532765293-30-7
    HIV-1 protease-IN-1 is a potent inhibitor of HIV-1 protease (IC50: 90 pM). HIV-1 protease-IN-1 has antiviral activity against B-HIV (EC50: 89 nM): HIV-1 protease-IN-1 was able to act on C-HIV strain ZM246 (EC50: 13.59 nM) and C-HIV strain Indie (EC50: 8.23 nM).
    • $2,140
    6-8 weeks
    Size
    QTY
    HIV-1 protease-IN-2
    T639492248124-46-9
    HIV-1 protease-IN-2 is a potent inhibitor of HIV-1 protease (IC50: 2.53 nM) and exhibits antiviral effects against DRV (Darunavir) sensitive and drug-resistant HIV-1 mutants.
    • $2,140
    6-8 weeks
    Size
    QTY
    HIV Protease Substrate I
    T76485124077-63-0
    HIV Protease Substrate I, a chromogenic substrate for HIV-1 protease, contains the protease's cleavage site [1].
    • Inquiry Price
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    HIV-1 protease-IN-8
    T789502925287-55-2
    HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme with an IC50 of 0.32 nM. It exhibits IC50 values of 0.29 μM for the wild-type HIV-1 (HIV-1 NL4-3) and 1.90 μM against a drug-resistant variant (HIV-1 MDR), indicating strong antiviral activity against both strains [1].
    • $1,970
    8-10 weeks
    Size
    QTY
    HIV-1 protease-IN-6
    T63733
    HIV-1 protease-IN-6 (compound 17d) is a potent HIV-1 protease inhibitor with an IC50 of 21 pM and a Ki of 4.7 pM, demonstrating significant antiviral activity against DRV (darunavir) resistant mutants, surpassing its inhibition efficacy against wild-type viruses.
    • $1,520
    10-14 weeks
    Size
    QTY
    HIV-1 protease-IN-4
    T74488
    HIV-1 protease-IN-4 (Compound II-22), a potent inhibitor of the HIV-1 protease, acts as a prodrug for atazanavir and significantly enhances its bioavailability in rat plasma, achieving a 5-fold increase in the area under the curve (AUC) and a 67-fold increase in concentration at 24 hours (C24) compared to oral administration of atazanavir alone [1].
    • Inquiry Price
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    HIV Protease Substrate IV
    T76511128340-47-6
    HIV Protease Substrate IV, a substrate for HIV (human immunodeficiency virus) protease, facilitates the measurement of HIV-1 protease activity [1].
    • Inquiry Price
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    HIV-1 protease-IN-10
    T79493
    HIV-1 protease-IN-10 (Compound 2) exhibits HIV-1 latency reversing activity (IC50: 0.22 μM), selectively binds to the PKCδ C1b domain (IC50: 0.69 μM), and demonstrates stability against esterase-mediated hydrolysis [1].
    • Inquiry Price
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    HIV-IN-4
    T604262408729-03-1
    HIV-IN-4 (Compound 12) is a potent inhibitor demonstrating significant anti-HIV activities [1].
    • $1,520
    6-8 weeks
    Size
    QTY