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Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TP2100L Avexitide acetate 2051593-46-3 98%
Avexitide acetate
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
T76279L1 Retatrutide sodium salt 98%
Retatrutide sodium salt
Retatrutide sodium salt is a potent triple agonist peptide for glucagon receptor (GCGR), glucose-dependent proinsulinotropic polypeptide receptor (GIPR), and glu...
TP1111L1 Tirzepatide sodium salt 98%
Tirzepatide  sodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.
T78097L Mazdutide acetate(2259884-03-0 free base) 98%
Mazdutide acetate(2259884-03-0 free base)
Mazdutide acetate is a potent co-agonist of glucagon-like peptide (GLP-1R) and glucagon receptor (GCGR), a gastrin-regulating hormone analog.Mazdutide acetate st...
T63909 GLP-1R agonist 3 2428640-18-8 98%
GLP-1R agonist 3
GLP-1R agonist 3 is a thickened imidazole derivative compound that is a potent agonist of GLP-1R. GLP-1R agonist 3 has shown research potential in diabetes.
T37890L GLP-1(28-36)amide acetate T37890L 98%
GLP-1(28-36)amide acetate
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
TP1863L Glucagon (19-29), human acetate TP1863L 98%
Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
T11408 Orforglipron 2212020-52-3 98%
Orforglipron
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1 diab...
TP1039 Secretin (33-59), rat 121028-49-7 98%
Secretin (33-59), rat
Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.
TP2252 GLP-1 (9-36) amide 161748-29-4 98%
GLP-1 (9-36) amide
antagonist at the human GLP-1 receptor
T76559 Survodutide 2805997-46-8 98%
Survodutide
Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor (GLP Receptor) that reduces body weight in HbA1c16 diabetes.
TP1111 Tirzepatide 2023788-19-2 98%
Tirzepatide
Tirzepatide (LY-3298176) is a dual agonist of glucose-dependent polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor with neuroprotective activity for ...
T40997 GLP-1R modulator C16 875005-43-9 98%
GLP-1R modulator C16
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
T40279 GLP-1R modulator L7-028 2648317-95-5 98%
GLP-1R modulator L7-028
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
T35337L Teduglutide acetate 98%
Teduglutide acetate
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
TP2100 Avexitide 133514-43-9 98%
Avexitide
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
T15387 GLP-1R Antagonist 1 488097-06-9 98%
GLP-1R Antagonist 1
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
T9579 GLP-1 receptor agonist 9 2401892-71-3 98%
GLP-1 receptor agonist 9
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
T19117 3-Deoxyglucosone 4084-27-9 98%
3-Deoxyglucosone
3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein a...
T61483 GLP-1R modulator C5 421578-93-0 98%
GLP-1R modulator C5
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study o...
Avexitide acetate
TP2100L
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
Retatrutide sodium salt
T76279L1
Retatrutide sodium salt is a potent triple agonist peptide for glucagon receptor (GCGR), glucose-dependent proinsulinotropic polypeptide receptor (GIPR), and glu...
Tirzepatide sodium salt
TP1111L1
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.
Mazdutide acetate(2259884-03-0 free base)
T78097L
Mazdutide acetate is a potent co-agonist of glucagon-like peptide (GLP-1R) and glucagon receptor (GCGR), a gastrin-regulating hormone analog.Mazdutide acetate st...
GLP-1R agonist 3
T63909
GLP-1R agonist 3 is a thickened imidazole derivative compound that is a potent agonist of GLP-1R. GLP-1R agonist 3 has shown research potential in diabetes.
GLP-1(28-36)amide acetate
T37890L
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
Glucagon (19-29), human acetate
TP1863L
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
Orforglipron
T11408
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1 diab...
Secretin (33-59), rat
TP1039
Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.
GLP-1 (9-36) amide
TP2252
antagonist at the human GLP-1 receptor
Survodutide
T76559
Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor (GLP Receptor) that reduces body weight in HbA1c16 diabetes.
Tirzepatide
TP1111
Tirzepatide (LY-3298176) is a dual agonist of glucose-dependent polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor with neuroprotective activity for ...
GLP-1R modulator C16
T40997
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
GLP-1R modulator L7-028
T40279
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
Teduglutide acetate
T35337L
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
Avexitide
TP2100
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
GLP-1R Antagonist 1
T15387
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).
GLP-1 receptor agonist 9
T9579
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
3-Deoxyglucosone
T19117
3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein a...
GLP-1R modulator C5
T61483
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study o...
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TargetMol