T11461 |
NE 52-QQ57
|
1401728-56-0
|
99.93%
|
|
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory activity.
|
TP1666L |
Kisspeptin-10, rat acetate(478507-53-8 free base)
|
TP1666L
|
99.92%
|
|
Kisspeptin-10, rat acetate is an endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).
|
T22027 |
AH-7614
|
6326-06-3
|
99.91%
|
|
AH-7614 (AH 7614) is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.
|
T2664 |
Timapiprant
|
851723-84-7
|
99.89%
|
|
Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).
|
T3176 |
APD597
|
897732-93-3
|
99.87%
|
|
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.
|
T3171 |
GSK137647A
|
349085-82-1
|
99.87%
|
|
GSK137647A (GSK 137647) is a selective FFA4 agonist.
|
T22591 |
ATC 0175 hydrochloride
|
510733-97-8
|
99.84%
|
|
ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affini...
|
T4626 |
TC-O 9311 free base
|
|
99.81%
|
|
TC-O 9311 is a potent GPR139 agonist.
|
T4566 |
Lodoxamide
|
53882-12-5
|
99.81%
|
|
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.
|
TN2077 |
(+/-)-Pinocembrin
|
68745-38-0
|
99.79%
|
|
(+/-)-Pinocembrin (NSC-43318), a natural product from axillary pines, is a GPR120 ligand that promotes wound healing in the HaCaT cell line.
|
T33452 |
ML192
|
460331-61-7
|
99.79%
|
|
ML192 (CID1434953) is a selective GPR55 ligand antagonist. ML192 is an inhibitor that inhibits β-arrestin transport, ERK1/2 phosphorylation, and PKCβII transloca...
|
T2528 |
Latanoprost
|
130209-82-4
|
99.78%
|
|
Latanoprost (Xalatan) is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with an ocular hypertensive effect.
|
T19700 |
IBC 293
|
306935-41-1
|
99.74%
|
|
IBC 293 is selective for GPR109B over niacin receptor GPR109A. IBC 293 is a highly selective agonist for GPR109B, a human orphan G-protein-coupled receptor expre...
|
T11458 |
GPR40/FFAR1 modulator 1
|
874755-26-7
|
99.72%
|
|
GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric modulator.
|
T10691 |
CAY10595
|
916047-16-0
|
99.71%
|
|
CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.
|
T3919 |
Ginsenoside Rb2
|
11021-13-9
|
99.66%
|
|
Ginsenoside Rb2 (Ginsenoside C) found in species of Panax, upregulating GPR120 gene expression.
|
T12375 |
Fezagepras sodium
|
1254472-97-3
|
99.59%
|
|
Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist or inverse agonist for GPR84, with anti-fibrotic, anti-inflamma...
|
T60184 |
TUG-499
|
1206629-08-4
|
99.59%
|
|
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 has an affinity for FFAR1 or GPR40 over the related receptors FFA...
|
T27850 |
LP-471756
|
413605-11-5
|
99.59%
|
|
LP-471756 is a specific antagonist of GPR139 and inhibits LP-360924-stimulated cAMP production (IC50 = 640 nM).
|
T15388 |
GLPG0974
|
1391076-61-1
|
99.58%
|
|
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
|