T78593 |
JP104
|
887264-45-1
|
98%
|
|
JP104 is an aryl carbamate that irreversibly inhibits fatty acid amide hydrolase (FAAH) with a pIC50 value of approximately 8 [1].
|
T78674 |
Isopropyl dodec-11-enylfluorophosphonate
|
623114-64-7
|
98%
|
|
Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibits equipot...
|
T16847 |
SA 47
|
792236-07-8
|
98%
|
|
SA 47 is a selective and effective inhibitor of fatty acid amide hydrolase and carbamate.
|
T12826 |
SA57
|
1346169-63-8
|
98%
|
|
SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).
|
T11255 |
FAAH-IN-1
|
1242441-47-9
|
98%
|
|
FAAH-IN-1 is a fatty acid amide hydrolase (FAAH) inhibitor, with IC50s of 145 nM and 650 nM for rat and human FAAH, respectively.
|
T63536 |
Dual FAAH/sEH-IN-1
|
2756099-59-7
|
99.89%
|
|
Dual FAAH/sEH-IN-1 is a dual inhibitor of sEH (soluble epoxide hydrolase) (IC50: 9.6 nM) and FAAH (fatty acid amide hydrolase) (IC50: 7 nM) with high affinity an...
|
T3215 |
JNJ-42165279
|
1346528-50-4
|
99.89%
|
|
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279...
|
T2684 |
JNJ-1661010
|
681136-29-8
|
99.8%
|
|
JNJ-1661010 (Takeda-25) is an effective and specific FAAH inhibitor (IC50: 10/ 12 nM for rat/human), shows >100-fold selectivity for FAAH-1 than FAAH-2.
|
T3354 |
BIA 10-2474
|
1233855-46-3
|
99.79%
|
|
BIA 10-2474 is a long-acting reversible inhibitor of fatty acid amide hydrolase (FAAH) that increases levels of the neurotransmitter anandamide in the central ne...
|
T2338 |
JZL195
|
1210004-12-8
|
99.78%
|
|
JZL195 is a selective and efficacious dual FAAH/MAGL inhibitor.
|
T8927 |
WWL 154
|
1338574-93-8
|
99.75%
|
|
WWL 154 is an serine hydrolase (SH) and fatty acid amide hydrolase FAAH-4 inhibitor.
|
T9374 |
AA38-3
|
65815-76-1
|
99.70%
|
|
AA38-3 (1-Piperidinecarboxylic acid, 4-nitrophenyl ester) inhibites three SHs (ABHD6, ABHD11, and FAAH)
|
T12139 |
N-(3-Methoxybenzyl)Palmitamide
|
847361-96-0
|
99.65%
|
|
N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders.
|
T4859 |
1-Monomyristin
|
589-68-4
|
99.58%
|
|
1-Monomyristin (2,3-Dihydroxypropyl tetradecanoate) , a 1-monoglyceride of myristic acid, has antibacterial activity against several Gram-positive bacterial stra...
|
T8646 |
URB937
|
1357160-72-5
|
99.55%
|
|
URB937 is an inhibitor of FAAH and increases anandamide levels(IC50 : 26.8 nM).
|
T67745 |
CB2R/FAAH modulator-2
|
2876918-68-0
|
99.52%
|
|
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH. CB2R/FAAH modulator-2 acts as a CB2R agonist and FAAH inhibitor, the Ki value...
|
T77513 |
2-Chlorophenylboronic acid
|
3900-89-8
|
99.42%
|
|
2-Chlorophenylboronic acid is a monohalogenated phenylboronic acid, which is an important pharmaceutical intermediate and is widely used in the synthesis of new ...
|
T77594 |
VU534
|
923509-20-0
|
99.22%
|
|
VU534 is a NAPE-PLD agonist with an EC50 of 0.30 μM.VU534 is a dual inhibitor of FAAH and sEH, with an IC50 of 1.2 μM for sEH.VU534 is used in diseases related t...
|
T15268 |
FAAH-IN-2
|
184475-71-6
|
99.18%
|
|
FAAH-IN-2 (O-Desmorpholinopropyl Gefitinib) is a potent inhibitor of FAAH(fatty acid amide hydrolase).
|
T7688 |
4-Nonylphenylboronic acid
|
256383-45-6
|
99.13%
|
|
4-Nonylphenylboronic acid is a inhibitor of FAAH.
|