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Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T8370 GSK5182 877387-37-6 97.63%
GSK5182
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
TN1768 Iriflophenone 52591-10-3 97.53%
Iriflophenone
Iriflophenone stimulates cells proliferation in  MCF-7 and T-47D human breast cancer.
T1571 Estriol 50-27-1 97.48%
Estriol
Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urina...
T0035 Dienestrol 84-17-3 96.73%
Dienestrol
Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the va...
T2250 DY131 95167-41-2 96.72%
DY131
DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.
T3645 Endoxifen E-isomer hydrochloride 1197194-61-8 96.47%
Endoxifen E-isomer hydrochloride
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
T1579 Mestranol 72-33-3 100%
Mestranol
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
T3846 Bavachin 19879-32-4 100%
Bavachin
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
T1424 Ethynyl estradiol 57-63-6 100%
Ethynyl estradiol
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is of...
T7389 G15 1161002-05-6
G15
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
T5633 H3B-5942 2052128-15-9
H3B-5942
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
T6743 (E/Z)-4-Hydroxytamoxifen 68392-35-8
(E/Z)-4-Hydroxytamoxifen
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeu...
T21897L MPP hydrochloride 98%
MPP hydrochloride
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
TN1567 Delphinidin chloride 528-53-0 98%
Delphinidin chloride
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of ...
T13542 α-Zearalenol 36455-72-8 98%
α-Zearalenol
α-Zearalenol is one of the major metabolites of Zearalenone. α-Zearalenol has structural analogy to estrogen, thus α-Zearalenol can bind to estrogen receptors (E...
T20625 Prochloraz 67747-09-5 98%
Prochloraz
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochlora...
GSK5182
T8370
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
Iriflophenone
TN1768
Iriflophenone stimulates cells proliferation in  MCF-7 and T-47D human breast cancer.
Estriol
T1571
Estriol (Oestriol) is a hydroxylated metabolite of ESTRADIOL or ESTRONE that has a hydroxyl group at C3, 16-alpha, and 17-beta position. Estriol is a major urina...
Dienestrol
T0035
Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the va...
DY131
T2250
DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.
Endoxifen E-isomer hydrochloride
T3645
Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
Mestranol
T1579
Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
Bavachin
T3846
Bavachin (Corylifolin) is a phytoestrogen that activates the estrogen receptors ERα and ERβ.
Ethynyl estradiol
T1424
Ethynyl estradiol is a semisynthetic alkylated ESTRADIOL with a 17-alpha-ethinyl substitution. It has high estrogenic potency when administered orally, and is of...
G15
T7389
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
H3B-5942
T5633
H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).
(E/Z)-4-Hydroxytamoxifen
T6743
(E/Z)-4-Hydroxytamoxifen (Afimoxifene) is the active metabolite of tamoxifen and a selective estrogen receptor (ER) modulator that is widely used in the therapeu...
MPP hydrochloride
T21897L
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
Delphinidin chloride
TN1567
Delphinidin chloride, a natural plant pigment found in berries and red wine, is a precursor of certain anthocyanins. Delphinidin chloride induces the release of ...
α-Zearalenol
T13542
α-Zearalenol is one of the major metabolites of Zearalenone. α-Zearalenol has structural analogy to estrogen, thus α-Zearalenol can bind to estrogen receptors (E...
Prochloraz
T20625
Prochloraz (Prelude) is a broad-spectrum contact imidazole fungicide. Prochloraz inhibits human placental microsomal aromatase in vitro (IC50 = 40 nM). Prochlora...
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TargetMol