Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

Cat. No.	Product name	CAS No.	Purity
TQ0311	GSK163090	844903-58-8	99.45%
TQ0311	GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).
T11463	GR 103691	162408-66-4	99.44%
T11463	GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 an...
T11011	Dexpramipexole dihydrochloride	104632-27-1	99.44%
T11011	Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agon...
T5S2059	Glaucine	475-81-0	99.42%
T5S2059	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T8959	OS-3-106	1580000-17-4	99.4%
T8959	OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.
T21432	Molindone	7416-34-4	99.37%
T21432	Molindone ((±)-Molindone) is a therapeutic antipsychotic used to treat schizophrenia by blocking the action of dopamine in the brain. molindone is often used in ...
TN1081	Hirsuteine	35467-43-7	99.36%
TN1081	Hirsuteine is a natural product. It non-competitively antagonizes nicotine-mediated dopamine release by blocking ion permeation through nicotinic receptor channe...
T16472	Pericyazine	2622-26-6	99.36%
T16472	Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to t...
T22530	6-Chloromelatonin	63762-74-3	99.36%
T22530	6-Chloromelatonin is a potent melatonin receptor agonist, a 5-methoxyindole compound that competes for the same presynaptic melatonin receptor sites in the rabbi...
T28167	NGB 2904	189060-98-8	99.35%
T28167	NGB 2904 is a potent and selective antagonist of dopamine D3 receptor (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4...
T0031L	Ziprasidone hydrochloride	122883-93-6	99.34%
T0031L	Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic acti...
T23232	Remoxipride hydrochloride	73220-03-8	99.32%
T23232	Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-adrenoce...
T0137	Mirtazapine	85650-52-8	99.3%
T0137	Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T12383	PD 168568 dihydrochloride	1782532-06-2	99.27%
T12383	PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
T7632	Veralipride	66644-81-3	99.21%
T7632	Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.
T12510	PNU-177864 hydrochloride	1783978-03-9	99.20%
T12510	PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor. PNU-177864 hydrochloride is structurally consistent with a ...
T6835	Fenoldopam mesylate	67227-57-0	99.19%
T6835	Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties. It lowers blood pressure through a...
T9228	Propionylpromazine hydrochloride	7681-67-6	99.17%
T9228	Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.
T0074L	Chlorprothixene hydrochloride	6469-93-8	99.16%
T0074L	Chlorprothixene hydrochloride (Truxal hydrochloride) brings strong blocking effects by blocking the 5-HT2 D1, D2, D3, histamine H1, muscarinic and alpha1 adrener...
T0719	Tetrabenazine	58-46-8	99.13%
T0719	Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake i...