T13245 |
UCSF924
|
1434515-70-4
|
98%
|
|
UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).
|
T12288 |
Odapipam
|
131796-63-9
|
98%
|
|
Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
|
T1476L |
Pramipexole dihydrochloride
|
104632-25-9
|
98%
|
|
Pramipexole dihydrochloride could be used to treat Parkinson disease.
|
T22921 |
LE 300
|
274694-98-3
|
98%
|
|
dopamine D1 receptor antagonist
|
T10611 |
Brexpiprazole S-oxide D8
|
2748605-29-8
|
98%
|
|
Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium labeled Brexpiprazole S-oxide. Brexpiprazole S-oxide is a main metabolite of Brexpiprazole. Brexpiprazole is...
|
T21360 |
Asenapine
|
65576-45-6
|
98%
|
|
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, dopamine receptor, and histamine receptor antagonist with antipsychotic effects that is used to tre...
|
TQ0175 |
Dexpramipexole
|
104632-28-2
|
98%
|
|
Dexpramipexole (KNS-760704, R-(+)-Pramipexole) is a neuroprotective agent and weak non-ergoline dopamine agonist.
|
TQ0140 |
Sumanirole maleate
|
179386-44-8
|
98%
|
|
Sumanirole maleate (U-95666E) is a highly selective full agonist of the D2 receptor (ED50: 46 nM).
|
T7341 |
Diclofensine
|
67165-56-4
|
98%
|
|
Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.
|
T9540 |
Phenelzine
|
51-71-8
|
98%
|
|
Phenelzine is an antidepressant and mania drug, which is a monoamine oxidase inhibitor. Its antidepressant effect is similar to that of niacinamide. It can reduc...
|
T11799L |
L-745870
|
158985-00-3
|
98%
|
|
L-745870 is a high-affinity and selective human dopamine D4 receptor antagonist (Ki: 0.43 nM). L-745870 has excellent brain penetration. It considerably weaker D...
|
T12476 |
Pimozide-d4
|
1803193-57-8
|
98%
|
|
Pimozide D4 is a deuterium labeled Pimozide.
|
T13463L |
Dihydrexidine
|
123039-93-0
|
98%
|
|
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.
|
T13898 |
SPD-473 citrate
|
161190-26-7
|
98%
|
|
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
|
T10908 |
CY 208-243
|
100999-26-6
|
98%
|
|
CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.
|
T12865 |
SCH-23390 maleate
|
87134-87-0
|
98%
|
|
SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM, r...
|
T13652 |
Dicarbine
|
17411-19-7
|
98%
|
|
Double carbene can be used for the study of schizophrenia and alcoholism. It can block dopamine receptors in various parts of the brain and prevent the reduction...
|
T68023 |
Tolnapersine
|
70312-00-4
|
98%
|
|
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
|
T10681 |
Cariprazine D6
|
1308278-67-2
|
98%
|
|
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).
|
TN1424 |
Bacopaside X
|
94443-88-6
|
98%
|
|
Bacopaside X (9.06 μM) showed binding affinity towards the D1 receptor.
|